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6-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyridine-2-carbonitrile
(1S,5R)-6-(cyclopropylmethyl)-3-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-methoxyphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
2-{1-[(4-fluorophenyl)methyl]-4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methylquinolin-2-amine
(1R,5S)-8-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-3,8-diazabicyclo[3.2.1]octane
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1,3-benzothiazole
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-4-methylpyrimidin-2-amine
N-(3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)-N-methylmethanesulfonamide
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
{[(3S,4R)-1-(4-ethoxybenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-methyl-3-[2-(methylamino)pyridine-3-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
2-[5-(1-acetylpiperidin-4-yl)-1-[(4-chlorophenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-4-(ethylamino)-5-methyl-N-(2-methylprop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(2-fluorophenyl)-5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(3,5-dimethylphenyl)-4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperazin-2-one
1-[(4-methoxyphenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2,5-dimethylbenzamide
2-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}ethan-1-amine
2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
1-[3-({[(5-chloro-2,3-dimethoxyphenyl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
1-(2-{4-[2-methyl-3-(2H-1,2,3,4-tetrazol-5-yl)pyridin-4-yl]phenyl}phenyl)ethan-1-one
2,3-difluoro-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
4-{1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-{[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,6-dimethoxyphenol
[3-(3-phenylpropyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-yl]methanol
(3R,4R)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
ethyl 2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)acetamide
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pyridine-3-carboxamide
4,6-dimethyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(1-benzylpyrrolidin-3-yl)-5-methyl-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
(2R)-2-hydroxy-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}propanamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[4-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
2-(8-fluoro-4-oxo-1,4-dihydroquinoline-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(pyrrolidin-3-yl)benzamide
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-[4-(methoxymethyl)piperidin-1-yl]acetic acid
2-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzoic acid
5-(2,2-dimethylpropanoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide