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(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
2-(1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-1,5-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(4-methoxyphenyl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-2-{[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
N-({1-[2-(4-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl 1-[(3R,5S)-1-(pyridin-2-ylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-(butan-2-yl)-3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-butyl-2-methyl-3-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
N-(1-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
1-(5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
1,9-dimethyl-4-[4-(methylamino)pyrimidin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
6-chloro-2-[2-(diethylamino)pyrimidin-5-yl]-N,N-dimethylquinoline-4-carboxamide
4-(2-methylphenoxy)-1-(oxane-4-carbonyl)piperidine
2-benzyl-9-[2-(methylamino)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aS)-5-[3-(1,3-benzothiazol-2-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-1-[2-(cyclohexylmethyl)morpholin-4-yl]propan-1-one
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
3-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2-[(3-methoxyphenyl)methyl]-4-(2,2,6,6-tetramethylpiperidin-4-yl)morpholine
{2-oxo-2-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}urea
1'-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(6-ethoxypyridin-3-yl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}oxan-4-amine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(furan-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-{[ethyl(2-hydroxyethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-acetyl-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[(3R,4S)-1-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-4-propylpyrrolidin-3-yl]ethane-1-sulfonamide
2-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)-1-methyl-1H-1,3-benzodiazole
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(ethanesulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-3-phenyl-1,2-oxazole
7-[(4-fluorophenyl)methyl]-2-(1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-cyclopropyl-N,4-dimethylpyrimidine-5-carboxamide
[(3S,5R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
4-(1-methyl-1H-pyrazol-4-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(methylsulfanyl)ethan-1-one
5-(2-{[(4,6-dimethylpyrimidin-2-yl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
2-methyl-5-[4-(3-methylphenoxy)piperidine-1-carbonyl]pyrimidine
(3R,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
methyl 4-{[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}butanoate
N-ethyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)furan-3-carboxamide