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4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-cyclohexyl-3-(furan-2-yl)-5-(methoxymethyl)-1H-1,2,4-triazole
6-amino-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyridine-3-carboxamide
1-(cyclopropylmethyl)-5-(2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S,4S)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-[methyl(2-methylpropyl)amino]pyrrolidin-3-ol
5-(2-{2-[(1,3-benzoxazol-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-2,3-dimethoxybenzamide
1-(1,4-dioxane-2-carbonyl)-4-[(2-methoxyphenyl)methyl]piperazine
N3-ethyl-4-oxo-1-(2-phenylethyl)-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
[(4-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1,3-thiazol-2-yl)methyl]dimethylamine
2-{[2-amino-6-(1-benzofuran-2-yl)pyrimidin-4-yl]amino}ethan-1-ol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][(1-phenyl-1H-pyrazol-4-yl)methyl]amine
5-{4-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}pyrimidine
4-(1,3-benzothiazol-2-yl)-N-(1-ethyl-1H-1,2,3-triazol-4-yl)-1,4-diazepane-1-carboxamide
1-({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
ethyl 1-(4-acetylbenzenesulfonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
[(4-ethyl-5-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
3-{[4-(3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}piperidin-1-yl)piperidin-1-yl]methyl}pyridine
2-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
2-(2-methoxyethoxy)-1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-[(2E)-3-phenylprop-2-en-1-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
2-(dimethylamino)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)benzamide
N-methyl-N-{2-[(thiolan-3-yl)amino]ethyl}methanesulfonamide
1-[(6-methylpyridin-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-cyclobutanecarbonyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidine
1-butyl-4-(3-cyclohexyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclohexyl-3-(oxan-4-yl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
6-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
4-methyl-2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-({4-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]phenyl}methyl)acetamide
1-cyclohexyl-3-[(dimethylcarbamoyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
(1R,7S)-3-tert-butyl-6-[3-(piperidin-1-yl)azetidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-imidazol-2-yl]-N-methylbenzene-1-sulfonamide
methyl 3-(cyclobutylmethoxy)-5-(3-oxopiperazine-1-carbonyl)benzoate
6-[methyl(1,2-oxazol-3-ylmethyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
5-methoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-oxo-1,4-dihydropyridine-2-carboxamide
1-ethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperidine-2-carboxamide
N-[3-(3-ethylphenoxy)propyl]-N-methyl-2-(2-oxoimidazolidin-1-yl)acetamide
4-methyl-6-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
N-{[1-(4-fluorophenyl)cyclopentyl]methyl}-1H-1,2,4-triazole-5-carboxamide
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2-cyclopentyl-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(propan-2-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-ethyl-1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-methylurea