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1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
3,4-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
2-(2-{[3-(methylcarbamoyl)pyrrolidin-1-yl]methyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
3-chloro-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-4-hydroxybenzamide
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
(1S,9R)-N-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
2-methyl-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazine-1,1-dione
2-(oxolan-2-ylmethyl)-9-(3-propyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-fluoro-3-methylphenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-{3-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-3-oxopropyl}piperidin-2-one
5-methoxy-1-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
2-{1-[1-(carbamoylmethyl)piperidin-4-yl]-N-methylformamido}-2-(pyridin-3-yl)acetic acid
N-(5-methyl-1,2-oxazol-3-yl)-2-{3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-{5-[(2-ethoxyphenyl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-({4-hydroxy-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]azepan-4-yl}methyl)thiophene-2-carboxamide
2-{5-cyclopropyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
2-benzyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
4-benzyl-3-ethyl-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-1,4-diazepan-5-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}benzamide
(1R,3S,5S)-8-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
3,6-dimethyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}morpholine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]methanol
N-methyl-2-(pyridin-3-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]pyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-benzyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-(3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-3-oxopropyl)-2-fluorobenzamide
3-cyclohexyl-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-5-(thiophen-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(4-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-[4-({[1-(cyclohexylmethyl)piperidin-3-yl]amino}methyl)phenyl]acetamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
methyl(oxolan-3-ylmethyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(1-phenoxypropan-2-yl)amine
4-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-yl]pyrimidine
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(2-methanesulfonylethyl)piperazine
(3S,4S)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N5-benzyl-N6-[2-methyl-2-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
6-{3-[4-(adamantan-1-yl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
3-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzonitrile
(2R,3R)-3-{[3-(1H-imidazol-1-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
N-[3-(2-methoxyphenyl)propyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-(cyclopropylmethyl)-8-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
(butan-2-yl)(3-phenylprop-2-yn-1-yl)(pyridin-4-ylmethyl)amine
4-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-phenylbutan-1-one