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(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{[2-(1H-pyrazol-1-yl)phenyl]methyl}cyclopentane-1,3-dicarboxamide
(2S,4R)-4-(dimethylamino)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxylic acid
methyl (2S,4R)-4-[4-(1H-pyrazol-1-yl)benzamido]-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
N-[(5-ethylpyridin-2-yl)methyl]-N,2-dimethylfuran-3-carboxamide
(1S,5R)-3-{[2-(difluoromethoxy)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aS)-2-propyl-5-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-1-(1-benzofuran-5-ylmethyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-[(2-chlorophenyl)methyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-methoxy-N-(1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(cyclopentylmethyl)-4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperazine
3-[1-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)piperidin-4-yl]-1,3-oxazolidin-2-one
methyl 5-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-methyl-2-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenol
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-5,8-dimethylquinolin-4-ol
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-2-(1H-pyrazol-1-yl)butanamide
N-[3-(dimethylamino)propyl]-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(morpholin-4-yl)-N-[3-(pyridin-2-yl)propyl]-2-(pyridin-3-yl)acetamide
2-[({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-6-methylpyridine-3-carbonitrile
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-phenoxyethan-1-one
2-{4-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]-1,4-diazepan-1-yl}-1,3-benzothiazole
N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl)methyl]acetamide
6-(3,4-dichlorobenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanamine
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
2-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
N4,6-dimethyl-N2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyrimidine-2,4-diamine
5-(4-{3H,3aH,4H,5H,9bH-cyclopenta[c]quinoline-4-carbonyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-{5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperidine
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(1-phenylethyl)-4H-1,2,4-triazole
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-methyl-5-{4-[4-(thiophen-2-yl)butanoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
6-(1-benzothiophene-5-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
1-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
2-[(4-chlorophenyl)methyl]-8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[(diethylamino)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
[(6-methoxypyridin-3-yl)methyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methoxyphenoxy)ethan-1-one
(3R,4R)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carboxamide
4-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-3-yl}pyrimidine
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide