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N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-cyclohexyl-3-methoxybenzamide
2,7-dimethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-5-methyl-1,3,4-oxadiazol-2-amine
1-[(5-acetylthiophen-3-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(2S)-4-methyl-1-oxo-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pentan-2-yl]acetamide
5-methyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1,3-oxazole-4-carboxamide
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
6-amino-N-[(3S,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]pyridine-3-carboxamide
3-{1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-5-[4-(1,3-thiazol-4-ylmethyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-methyl-1-[(4-methylphenyl)amino]-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]cyclopentane-1-carboxamide
N-{3-[2-(3,4-dichlorophenyl)morpholin-4-yl]propyl}methanesulfonamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
(2S)-2-{2-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}propanamide
1-[4-(2-hydroxyethyl)piperazin-1-yl]-3-(2-methylphenyl)-3-phenylpropan-1-one
1-methyl-1'-(morpholine-4-sulfonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
[7-(2,4-difluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1H-pyrrole-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-phenoxybenzamide
5-(1H-imidazol-1-ylmethyl)-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
1-[(2-chlorophenyl)methyl]-N-(quinolin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-(oxolane-3-carbonyl)piperazine
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
2-(cyclohexylmethyl)-4-(propane-1-sulfonyl)morpholine
N-cyclohexyl-2-(4-methanesulfonamidopiperidin-1-yl)butanamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-({3-carboxy-4H,5H,6H,7H-thieno[2,3-c]pyridin-2-yl}sulfonyl)piperidine-4-carboxylic acid
(4aS,7aR)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-3-methyl-N-propylbenzamide
2-methyl-3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
4-(2-ethoxyphenyl)-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-1-ene-1-carboxamide
2-(2-ethoxypyridin-3-yl)-3-(pyrrolidine-1-carbonyl)pyridine
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(2-phenylethyl)piperidine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-[(3S,4R)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-methyl-4-phenyl-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
6-methyl-3-[(3-phenylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-cyclopentyl-5-[1-(furan-3-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3-difluoro-4-methoxy-N-(2-methoxyethyl)benzamide
1,2-dimethyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indol-5-ol
N-methyl-N-(2-phenylethyl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-amine
(1-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol