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2-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
propan-2-yl 4-{[3-(3-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(1R,7S)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-tert-butyl-7,7-dimethyl-N-[(6-methylpyridin-2-yl)methyl]-5,6,7,8-tetrahydroquinazolin-5-amine
2-(morpholin-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2-(pyridin-3-yl)acetamide
(3aS,6aS)-2-[(4-chloro-3-fluorophenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aR,7aS)-2-{2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-{4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-[3-(4-fluorophenyl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}phenol
5-{2-[3-(oxolan-3-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
3-hydroxy-N-(2-methyl-1-benzofuran-5-yl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
2,6-dimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-4-carboxamide
5-ethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-{2-[4-(3-methyl-1-benzofuran-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}pent-4-en-1-one
3-cyclopropyl-1-phenyl-N-(1,3-thiazol-2-yl)-1H-1,2,4-triazole-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
{[2-ethoxy-5-(isoquinolin-5-yl)phenyl]methyl}(methyl)amine
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
4-[(2-methylprop-2-en-1-yl)oxy]-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)benzamide
4-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}-N-(pyridin-4-yl)benzamide
methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
N-(1-methanesulfonylpiperidin-4-yl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-{3-[(4-methoxyphenyl)methyl]-5-(1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
N,N-dimethyl-2-{2-[4-(pyridin-2-yl)phenyl]-1H-imidazol-1-yl}ethane-1-sulfonamide
(4-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
7-(1,3-benzothiazol-2-yl)-4-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-cyclopropyl-1-(propan-2-yl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
N1-(3-fluoro-5-methylphenyl)-N4-(1-methoxypropan-2-yl)piperidine-1,4-dicarboxamide
2-(2-chloro-4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenoxy)acetamide
5-oxo-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-dihydroquinolin-2-one
1-cyclopentyl-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazin-2-one
N-[3-(1H-pyrazol-1-yl)propyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
5-[(dimethylamino)methyl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazole-2-carboxamide
1'-[4-(1H-imidazol-1-yl)butanoyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-acetamido-N-[4-(furan-2-ylmethoxy)phenyl]pyrrolidine-1-carboxamide
4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-(dimethyl-1,2-oxazole-4-carbonyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-3-(2-oxoazepan-1-yl)propanamide
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-5-methylphenol
4-methyl-2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrrole
3-(5-oxo-1-propylpyrrolidin-3-yl)-1-[3-(piperidine-1-carbonyl)phenyl]urea
N-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-yl}-N-methylacetamide
(1S,6R)-9-{[2-(methylamino)pyridin-3-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-chloro-5-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}amino)-N-propylbenzamide
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
5-methyl-3-(4-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}phenyl)-1,2,4-oxadiazole