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4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxolan-3-yl)-1H-pyrazole-3-carboxamide
N-benzyl-5-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(prop-2-en-1-yloxy)phenyl]urea
N-[3-(4-chlorophenyl)propyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
(1R,3S,4S)-3-hydroxy-4,7,7-trimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]bicyclo[2.2.1]heptane-1-carboxamide
3-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-ethyl-N-methyl-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-{4-[1-(morpholin-4-yl)ethyl]phenyl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
3-[5-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidin-4-amine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[2-(5-methylfuran-2-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
11-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-4-(1H-pyrazol-3-yl)benzamide
2-(3-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
{8-methyl-2-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]quinolin-3-yl}methanol
14-(5-butylthiophen-2-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(1-methoxypropan-2-yl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-fluorophenyl)-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{4-[(2-aminopyridin-3-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
3-(2-fluoro-5-methanesulfonamidophenyl)-1-[(3-hydroxypiperidin-3-yl)methyl]urea
1-{5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
8-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-[(2-hydroxy-6-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N,1-dimethyl-2-oxo-6-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[2-(2-methyl-1H-indol-3-yl)acetyl]piperidine-3-carboxylic acid
3-{[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]amino}-N-(pyridin-3-yl)propanamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
N-benzyl-N-[2-(dimethylamino)ethyl]-1-[2-(2-methoxyethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
4-chloro-1-methyl-3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}-1H-indazole
3-[3-({[2-(morpholin-4-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(5-methyl-1H-pyrazol-1-yl)propanamide
(1S,5R)-N-(2,4-difluorophenyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
(2S)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-chloro-N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-[(2,3,5,6-tetrafluoro-4-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
(2S,4R)-4-amino-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-N,N-diethylpyrrolidine-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
N-{3-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]propyl}pyridine-4-carboxamide
3-cyclopropyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
3-(2-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
4-{5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol