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1-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-4-yl)-2-phenylethan-1-ol
3-[(4aR,8aR)-6-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-(2,3-dimethoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
1-(2H-1,3-benzodioxol-5-yl)-N,N-diethyl-3-(2-methylpropyl)-1H-1,2,4-triazole-5-carboxamide
2-methyl-1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indole-3-carbonitrile
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}quinoxaline
5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}quinoxaline
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(dimethylamino)-7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-methyl-6-[4-({[3-(pyrrolidin-1-yl)phenyl]methyl}amino)piperidin-1-yl]pyrimidin-2-amine
1,9-dimethyl-4-[(2-propoxyphenyl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
3-cyclopropyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-{methyl[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}propane-1,2-diol
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(pyridin-3-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{[4-(3-chloropyridin-2-yl)piperazin-1-yl]methyl}benzoic acid
(1S,5R)-3-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(4-fluorophenoxy)ethan-1-one
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{3-methyl-1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-(propan-2-yl)-1H-pyrazole
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-(3-methylphenyl)piperidine
2-{4-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazin-1-yl}ethan-1-ol
N-benzyl{[2-(morpholin-4-yl)phenyl]amino}sulfonamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
4-(piperidin-3-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
N-[(2S)-1-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1-oxopropan-2-yl]acetamide
1-tert-butyl-4-[({5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)methyl]pyrrolidin-2-one
8-[5-(trifluoromethyl)pyridin-2-yl]-1-oxa-8-azaspiro[4.5]decane
5-cyclobutyl-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-1,3,4-oxadiazol-2-amine
2-[4-(4-ethylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
2-[(4aR,7aS)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-{4-[(2,3-difluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-methoxybenzoyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
methyl 5-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
[(3R,4R)-1-(1H-indole-6-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-benzyl-N-methyl-1-{2-[3-(pyridin-3-yl)propanamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(3-hydroxypropyl)phenyl]-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
4-[4-(2-methoxyphenyl)phenyl]-4H-1,2,4-triazole
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-methoxyethyl 1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxylate
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-[(2-methylphenyl)methyl]acetamide
6-{1-azabicyclo[3.2.1]octan-5-yloxy}-1,2,3,4-tetrahydronaphthalen-1-one
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrrole-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
1-{2-hydroxy-3-[2-methoxy-4-(piperidin-1-ylmethyl)phenoxy]propyl}piperidin-4-ol
3-{2-oxo-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)(pyridin-4-ylmethyl)amine
N-[4-(3-methoxyphenyl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide