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N-[(2,4-dihydroxyphenyl)methyl]-3-(2-fluorophenyl)-3-phenylpropanamide
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[4-(thiophene-3-carbonyl)morpholin-3-yl]acetamide
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-N,N-dimethylpyrrolidine-2-carboxamide
7-[1-(2-fluorophenyl)cyclopropanecarbonyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-[4-(dimethylamino)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{1-cyclohexyl-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(3-methoxyphenyl)-1-methyl-1H-imidazole
1-(4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(pyridin-3-yloxy)piperidine-1-carboxamide
(3aR,7aS)-2-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
4-[1-(3-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazole-5-carbonyl]morpholine
6-methyl-1-{3-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
N-[3-(methylsulfanyl)phenyl]-4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carboxamide
2,2-dimethyl-N-[1-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(2-hydroxyethyl)-3-(naphthalen-2-yl)prop-2-ynamide
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
7-(2-oxo-1,3-oxazolidin-3-yl)-4-(quinoxalin-2-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-{1-[2-(methylamino)pyridine-4-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethan-1-one
4-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-2-(trifluoromethyl)morpholine
1-(dimethylamino)-3-(2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-4-methoxyphenoxy)propan-2-ol
4-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-(2-oxoimidazolidin-1-yl)benzamide
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-N-methylpyridin-2-amine
1-[2-(4-methylpentyl)morpholin-4-yl]-3-(methylsulfanyl)propan-1-one
4-(5-{[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
3-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
(1S,4S)-2-(2-fluorophenyl)-5-{[4-(trifluoromethyl)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
4-cyclobutyl-6-methyl-N-[1-(6-methylpyridin-2-yl)propyl]pyrimidin-2-amine
4-ethyl-1-(2-hydroxyethyl)-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[2-(2-aminoethyl)morpholin-4-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-(2-{[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}ethyl)acetamide
2-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,3-dihydroxy-2-methylpropan-2-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2-ethylphenyl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
6-[4-(pyrrolidine-1-carbonyl)phenyl]pyridin-2-amine
2-(3-methoxypropyl)-8-(4-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
4-{5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
6-(2-fluoro-4-methoxyphenyl)-N-(2-hydroxyethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)cyclopropan-1-amine
3-{1-[2-(4-chlorophenoxy)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol