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1-{3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-3-methoxypiperidine
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-methylpropan-1-one
(2S,4R)-4-{[(2-chlorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-cyclohexyl-3-{[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}propanamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
(3E)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pent-3-en-1-one
2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}-2-[4-(methylsulfanyl)phenyl]acetic acid
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-methylprop-2-en-1-yl)amine
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl]methanol
N-(2-fluorophenyl)-4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-3-(3-{1-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-amine
4-[(2-ethoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
3-({3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)pyridine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]pyridine-4-carboxamide
N-[4-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
7-amino-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-1-(2-methoxyacetyl)piperidine-3-carboxamide
4-{2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}piperazine-2-carboxylic acid
1-methoxy-8-[2-(4-phenylphenyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
8-(2-methylfuran-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-[(4-chloro-3-fluorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(ethylamino)-N-[(2-fluorophenyl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(pyrrolidin-3-yl)pyridin-2-amine
1-{3-[(2,2-dimethylpyrrolidin-1-yl)methyl]phenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5-methylpyrazine
1-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]-2-phenylethan-1-one
1-(2-chloro-6-methylphenyl)-3-cyclopentyl-3-[2-(dimethylamino)ethyl]urea
1-(1,3-benzothiazol-2-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidin-4-amine
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
propan-2-yl 4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}piperidine-1-carboxylate
N4-[(1-benzylpiperidin-4-yl)methyl]-N4-methylpyrimidine-2,4,6-triamine
N-[(3-chlorophenyl)methyl]-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
1-(1-methyl-3-propyl-1H-pyrazole-5-amido)cyclopentane-1-carboxylic acid
methyl 4-{[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]methyl}benzoate
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-amino-4-(3-ethyl-1,2-oxazol-5-yl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
4-phenyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carbonitrile
4-hydroxy-1-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]piperidine-4-carboxylic acid
3-cyclobutyl-4-(1H-indol-4-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-phenylpropyl)morpholine