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1-benzyl-N,N-dimethyl-5-{[4-(2-methylpropyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(pyrrolidin-3-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
(3S,4R)-4-(3-fluorophenyl)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxylic acid
2,6-dimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinoline-4-carboxamide
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)methylamine
methyl(2-phenoxyethyl)(pyridin-2-ylmethyl)amine
(4aS,7aR)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-4-[({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)methyl]pyrrolidin-2-one
N-[(3S,4R)-1-(4-phenoxybutanoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(furan-2-ylmethyl)-2-(4-methyl-1,4-diazepan-1-yl)-N-(thiophen-2-ylmethyl)acetamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-(1H-pyrazol-3-yl)benzamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane-6-carboxylic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
methyl 6-(1-methoxypropan-2-yl)-2-{[(4-methylphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
8-[(2,4-dimethylphenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(furan-2-yl)-3-phenylpropan-1-one
(3S,4R)-1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
1,5-dimethyl-2-phenyl-4-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)-2,3-dihydro-1H-pyrazol-3-one
1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
2-(1,2-benzoxazol-3-yl)-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
7-methyl-2-(pyrimidin-5-yl)-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
7-(2-hydroxyethyl)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,7-diazaspiro[4.5]decan-6-one
2-(2-{[2-(pyridin-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
propyl(pyridin-3-ylmethyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
3-ethyl-4-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazin-2-one
N-[2-(pyridin-3-yloxy)propyl]-1H-imidazole-2-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}acetamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(2-acetylphenyl)-N-(propan-2-yl)benzamide
2-(2-ethoxypyridin-3-yl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
2-ethyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 4-{[(1S,4S)-5-[2-(methylsulfanyl)phenyl]-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}benzoate
2-[benzyl({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
4-(2H-1,3-benzodioxol-5-yl)-2-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}phenol
3-{3-[4-(1-ethyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]propyl}pyridine
ethyl 1-{1-[2-(benzenesulfonyl)ethyl]-7-oxoazepan-4-yl}piperidine-2-carboxylate
4-(propan-2-yl)-6-(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine-1-carbonyl)pyrimidin-2-amine
4-[(3aR,6aR)-2-benzyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-1,4-diazepan-2-one
N-propyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyridine-3-carboxamide
2-(2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
1-methyl-4-(oxan-4-yl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N4-[(6-chloropyridin-3-yl)methyl]-N4,N6,N6-trimethylpyrimidine-4,6-diamine