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1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
2-(4-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}piperazin-1-yl)ethan-1-ol
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[4-(pyrrolidin-1-ylmethyl)phenyl]methyl})amine
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
1-[(2-chloro-4-fluorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-cyclopentyl-4-{2-[3-(methylamino)propoxy]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(3-chlorophenyl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidine-3-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
ethyl 2-[({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]acetate
(1R,6S)-9-methyl-3-(1H-pyrrole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-{[4-(3-methylpyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
3-{1-[2-(1H-pyrazol-1-yl)butanoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-[(5-methylthiophen-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
methyl 2-(ethylsulfamoyl)-6-[2-(methoxycarbonyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
(1H-indol-5-ylmethyl)(2-methoxyethyl)(thiophen-2-ylmethyl)amine
2-cyclopropyl-4-methyl-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidine
(cyclobutylmethyl)[(1,4-dimethyl-1H-pyrazol-5-yl)methyl](oxolan-2-ylmethyl)amine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{1-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N3-butyl-1-cyclopentyl-N3-methyl-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]acetamide
4-(4-fluorophenoxy)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
4-(4-chlorophenyl)-1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-ol
1-cyclopentyl-4-({[(3,5-dichloropyridin-4-yl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-(2-methylphenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
1-phenyl-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine
2-(carbamoylamino)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
N-(2,2-difluoroethyl)-4-[(2-methyl-1,4-oxazepan-4-yl)sulfonyl]benzamide
5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[5-(2-ethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
ethyl 4-{6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carbonyl}piperazine-1-carboxylate
(1R,3R)-N1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]cyclopentane-1,3-diamine
1-(furan-3-carbonyl)-3-(4-phenoxybenzoyl)piperidine
3-{1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-imidazol-2-yl}benzonitrile
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(1S,5R)-3-[5-(ethylsulfanyl)thiophene-2-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{2,2-dimethyl-3-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperazin-1-yl]propyl}dimethylamine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-indole-7-carboxamide
{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
(4aR,7aS)-1-(2,2-dimethylpropanoyl)-4-(3-fluorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-6-cyclobutanecarbonyl-4-(1H-indol-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2R,6R)-4-[(1-ethyl-1H-imidazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[5-(3-cyclohexyl-1H-pyrazol-4-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
2-{3-[7-(cyclopropylmethyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}pyridin-3-ol