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N'-(3-hydroxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)butanediamide
3-(1-2,3-dihydro-1H-inden-5-yl-N-methylformamido)-N-methylbutanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(propan-2-yloxy)acetyl]pyrrolidin-3-yl]pyridine-4-carboxamide
1-methyl-6-(pyridin-4-yl)-N-[2-(pyrrolidin-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,2S,6R,7S)-4-[4-(morpholine-4-carbonyl)benzoyl]-4-azatricyclo[5.2.2.02,6]undecane
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-methyl-N-[2-(piperidin-1-yl)ethyl]cyclopropane-1-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]propanamide
N-[(3-chlorophenyl)methyl]-3-{1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-yl}propanamide
2-{[(2-butyl-1H-imidazol-4-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-1H-indol-1-yl]propanamide
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-[2-(methylsulfanyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aS,8aR)-6-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
4-{4-[3-(furan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methoxypyrimidine
2-({[2-(dimethylamino)-2-(furan-2-yl)ethyl]amino}methyl)-8-fluoroquinolin-4-ol
(3aS,6aS)-2-(cyclopropylmethyl)-5-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
ethyl 4-[1-(6-cyanopyridin-2-yl)piperidin-3-yl]piperazine-1-carboxylate
methyl({[1-({1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl})amine
6-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-{3-[(pyridin-3-ylmethyl)carbamoyl]piperazin-1-yl}-1,3-oxazole-4-carboxylic acid
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
4-{2,8-dimethyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl}-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(3,4-dimethylphenoxymethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-{[(2-fluorophenyl)methyl](methyl)amino}-N-[(1-methylpiperidin-3-yl)methyl]acetamide
(1S,5R)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(1,3-benzoxazol-2-yl)piperidin-4-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-1-methyl-6-oxo-N-(thiophen-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxamide
1-(2-fluorophenyl)-3-(4-methoxyphenyl)-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
[(3R,4R)-1-(3,4-difluorobenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(1H-imidazol-1-yl)-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
1-({5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-(3-methylbenzoyl)pyrrolidine-2-carboxamide
N-methyl-4-[2-oxo-2-(piperidin-1-yl)ethoxy]-N-(1H-pyrazol-5-ylmethyl)benzamide
1-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-3-(4-methoxy-2-methylphenyl)urea
1-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
4-{2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]ethyl}benzoic acid
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}[(1-ethyl-1H-imidazol-5-yl)methyl]amine
2-[(1S,5R)-3-[(2-fluoro-5-methoxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
(1R)-2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-phenylethan-1-ol
7-fluoro-4-[2-(furan-2-yl)azepane-1-carbonyl]-2-methylquinoline
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-5-propyl-1,3,4-oxadiazol-2-amine