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(2S,4R)-4-amino-N-(propan-2-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidine-2-carboxamide
1'-(1-methyl-1H-imidazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3R,4R)-3-hydroxy-1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]pyridine-4-carboxamide
methyl 2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
2-methyl-2-{4-[3-(methylamino)pyrazin-2-yl]phenyl}propanenitrile
7-(2-methoxyethyl)-2-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-chloro-2-ethylphenyl)-3-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
2-(4-fluorophenyl)-N-(2-hydroxyethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-{[7-(2-methoxy-2-phenylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-indole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
methyl 3-(1-benzothiophen-2-ylmethyl)-9-(cyclopentyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(3-chloro-4-fluorobenzoyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
N-[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]methanesulfonamide
4,5-dimethyl-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidine
3-(2-methoxy-5-methylphenyl)pyridin-2-ol
(3aS,7aR)-2-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,5R)-3-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,9-diazabicyclo[3.3.2]decan-10-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}piperidin-2-one
2-(adamantan-1-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
(2S)-4-[(3,5-dimethyl-1H-indol-2-yl)formamido]-2-hydroxybutanoic acid
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-(4-cyanophenyl)-4-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]butanamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2-methoxyethyl)-8-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4S)-4-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1,4-diazepan-1-yl]oxolan-3-ol
2-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-4-methyl-1,4-diazepane-1-carboxamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-(2,2-diphenylethyl)-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3,5-dimethyl-N-{[4-(morpholin-4-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
1-[1-(furan-2-yl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]urea
[7-(isoquinolin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoacetamide
[(2-fluoro-5-methoxyphenyl)methyl](methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(thiomorpholin-4-yl)propan-1-one
6,7-dimethyl-2-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1H-1,3-benzodiazole
2-cyclopropyl-4-phenyl-9-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane
3-[({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}carbamoyl)methyl]-1,2,3-oxadiazol-3-ium-5-olate
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
methyl[2-(oxan-4-yl)ethyl][(2,3,4-trifluorophenyl)methyl]amine
{2-[4-(2-amino-1H-imidazol-5-yl)phenyl]phenyl}methanol
4-methyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-oxazole-5-carboxamide
(1R,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(5-methylfuran-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-3-(2-methylphenyl)pyrrolidin-3-ol