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2-(2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
3-(azepane-1-carbonyl)-1-ethyl-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(azocan-1-yl)-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)propanamide
3-[(2-chloro-4-fluorophenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(6-methylpyridin-2-yl)piperazine
N-(2-fluorophenyl)-3-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
4-[(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
(4aS,7aR)-1-(2,5-difluorobenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
2-[3-(3-chlorophenoxymethyl)-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
(1R,3S,5S)-N-benzyl-3-hydroxy-8-azabicyclo[3.2.1]octane-8-sulfonamide
4-(5,6-dimethylpyridine-3-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
3-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole
3-methyl-7-[2-(4-propoxyphenoxy)ethyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-cyclopropylpropanamide
N,6-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-{[1-(4-fluorophenyl)cyclopentyl]methyl}-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
8-(2,8-dimethylquinoline-4-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
5-(2-methoxyquinolin-3-yl)-3-methylpyridin-2-amine
4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
3-{1-[2-(3-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
1-(3-{[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]amino}propyl)pyrrolidin-2-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
N-[2-(methylsulfanyl)phenyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
1-ethyl-4-{[methyl({6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl})amino]methyl}pyrrolidin-2-one
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(4-methoxyphenyl)-2-methylpiperazine
3-fluoro-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
methyl 2-chloro-4-{[(oxolan-2-ylmethyl)(propyl)carbamoyl]amino}benzoate
3-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
2-(5-methyl-1,2-oxazol-3-yl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
3-(5-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
6-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]pyrazine-2-carboxamide
3-(2-methanesulfonamidoethyl)-1-(2-methyl-1-benzofuran-5-yl)urea
N,5-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-{3-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]phenoxy}acetamide
5-{8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-[(2,3-difluorophenyl)methyl]-2-(3-methoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[3-(hydroxymethyl)quinolin-2-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(2-methyl-6-{1-[2-(oxolan-3-yl)ethyl]piperidin-4-yl}pyrimidin-4-yl)morpholine
methyl 4-({5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)butanoate
3-cyclopropyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{2-[methyl(phenyl)amino]propyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N,N-dimethyl-2-({2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide