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1-(2-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
6-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-fluorobenzamide
(3R,4R)-1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-fluoro-5-(3-methoxypiperidine-1-carbonyl)phenol
3-[1,5-dimethyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-N,N-dimethylbenzamide
4-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,5-dimethylpyrimidine
3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[2-(2-methylphenyl)ethyl]amine
methyl 6-[(2-hydroxyphenyl)methyl]-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl[2-(1-methylpiperidin-4-yl)ethyl]{[2-(trifluoromethyl)phenyl]methyl}amine
(1R,7S)-3-cycloheptyl-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(5-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]pyrazolo[1,5-a]pyridine-7-carboxamide
5-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(5-acetamido-2-methylphenyl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
4-(3-chloro-5-fluoro-4-methoxyphenyl)-1-(1,4-dioxan-2-ylmethyl)-1H-1,2,3-triazole
[7-(2-methyl-1H-imidazol-4-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methanamine
7-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[3-(phenylsulfanyl)propyl]pyrimidin-2-amine
1-(2,5-dimethylfuran-3-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
9-(3-fluoropyridin-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cycloheptyl-2-methyl-N-(pyridin-3-ylmethyl)-5-sulfamoylbenzamide
3-methyl-5-(4-methylthiophen-3-yl)-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[(3S,4R)-4-(propan-2-yl)-1-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}pyrrolidin-3-yl]acetamide
2-(dimethylamino)-7-[2-(methylsulfanyl)pyridine-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[7-(cyclopent-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
[(2S,4R)-1-[(2E,4E)-5-(4-chlorophenyl)penta-2,4-dien-1-yl]-4-(dimethylamino)pyrrolidin-2-yl]methanol
3-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-(pyrrolidin-1-yl)propan-1-one
8-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
7,7-dimethyl-2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-6-methylphenol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(9H-purin-6-yl)piperidin-4-amine
3-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
2-methyl-2-[4-(morpholin-4-yl)-2-[4-(propan-2-yl)piperazin-1-yl]pyrimidin-5-yl]propanoic acid
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
3-[5-(2,6-dimethylquinoline-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
6-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}naphthalen-2-ol
1-cyclopentanecarbonyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
9-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(hydroxymethyl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-3-ol
methyl 6-[2-(3-fluorophenyl)acetyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-chloro-N,N-diethyl-3-({[2-(1,3-thiazol-2-yl)ethyl]carbamoyl}amino)benzamide
3,5-dimethoxy-2-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)benzoic acid
2-methyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N'-cyclooctyl-N-(2-methanesulfonylethyl)butanediamide
N-benzyl-4-(3-methoxyphenyl)-2-methyl-3-oxopiperazine-1-sulfonamide