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methyl 2-(ethylsulfamoyl)-6-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-phenyl-3-{1-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methoxy-N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-amino-N-methyl-N-[3-(oxolan-2-yl)propyl]cyclopropane-1-carboxamide
1-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-amino-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-methyl-1,3-thiazole-5-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[2-(methylsulfanyl)ethyl]benzamide
(3R,5R)-5-(morpholine-4-carbonyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)piperidine-3-carboxamide
2-(pyridin-2-yl)-7-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2,6-dimethyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]quinoline-3-carboxamide
(2R,6S)-4-[1-(2-ethoxypyridine-3-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
2-(dimethylamino)-2-(4-fluorophenyl)-1-(thiomorpholin-4-yl)ethan-1-one
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-(2-methylfuran-3-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
(1R,5R)-6-[(5-propylfuran-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
4-{[4-methyl-5-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
(cyclohexylmethyl)(methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-benzyl-8-[2-(methylsulfanyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(phenylsulfanyl)ethan-1-one
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
4-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
1'-[(4-methanesulfonylphenyl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
{[2-(azocan-1-yl)pyridin-3-yl]methyl}(furan-3-ylmethyl)amine
4,4-difluoro-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-[4-(2-methoxypyridin-3-yl)phenyl]ethan-1-ol
5-acetyl-2,4-dimethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1H-pyrrole-3-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,3-diphenyl-1H-pyrazole
4-(3-hydroxy-3-methylbutyl)-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]benzamide
N-cyclopropyl-4-methoxy-2-{[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]oxy}benzamide
(1R,2S,6R,7S)-4-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-4-azatricyclo[5.2.2.02,6]undecane
(3S,4R)-4-(2-methoxyphenyl)-1-(quinolin-4-ylmethyl)pyrrolidine-3-carboxylic acid
2-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-3-phenylcyclopent-2-en-1-one
3-(1-methylpiperidin-2-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]propanamide
(2R)-2-amino-N,4-dimethyl-N-[(5-methylfuran-2-yl)methyl]pentanamide
N4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(4-methoxy-2-methylphenyl)-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propanamide
methyl 4-({2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}carbamoyl)butanoate
1-{3,5-dimethyl-4-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)naphthalene-1-carboxamide
4-(pyridin-2-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
5-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
(3R,4R)-1-[(2-methyl-1-benzothiophen-3-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
1'-[(5-ethylpyridin-2-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]