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2-(1H-indol-3-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-{[(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(4-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}piperazin-1-yl)-2,2-dimethylpropan-1-one
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyridine-2-carboxamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-(furan-2-ylmethyl)piperidine
(2S,4R)-4-amino-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}(4,4,4-trifluorobutyl)amine
2-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-8-methoxyquinoline
3-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
(2R,5R)-N-(2-methoxy-6-methylphenyl)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazine-1-carboxamide
N-{4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]phenyl}ethane-1-sulfonamide
4-{1-[(dimethylcarbamoyl)methyl]piperidin-3-yl}benzoic acid
{[(3S,4R)-1-(2-fluoro-6-methoxybenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-amino-4-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
methyl 4-methoxy-3-{[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]methyl}benzoate
4-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-4-yl}pyrimidine
8-fluoro-2-[({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]quinolin-4-ol
[(3aS,6aS)-2-(2-ethylpyrimidine-5-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
9-(2-chloro-3-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-1-benzyl-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
2-(2-phenyl-1,3-thiazol-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N-(3-ethoxypropyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-[(5-methylthiophen-2-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(3aS,6aR)-5-[(2-methoxypyrimidin-5-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxypyridine-4-carboxamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
N-[(1S,2R)-2-aminocyclobutyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]propan-1-one
2-[(2-aminopyridin-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(6-aminopyridin-3-yl)-2-{4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}acetic acid
1-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
ethyl 4-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}piperidine-1-carboxylate
2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,3-thiazole-4-carboxamide
2-{[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]sulfanyl}pyridine
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-{2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-(3-chlorophenyl)-4-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperazin-2-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
2-methoxy-N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
4-[3-fluoro-5-(propan-2-yloxy)phenyl]-5-(methoxymethyl)-3-methyl-1H-pyrazole
3-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[(2-phenylpropan-2-yl)amino]methyl}piperidin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3-chlorophenyl)methyl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[(2-chloro-4-fluorophenyl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(oxolane-2-carbonyl)-1,4-diazepane
2-[3-phenyl-5-(piperidin-1-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine