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(2,1,3-benzoxadiazol-5-ylmethyl)[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-(morpholin-3-yl)acetamide
2-(4-phenylpiperazine-1-carbonyl)-3-(piperidine-1-carbonyl)pyrazine
3-[(6-chloropyridin-3-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-{[(3S,4S)-3-hydroxy-1-[2-(2-hydroxyphenyl)acetyl]piperidin-4-yl]methyl}cyclopentanecarboxamide
2-{1-cyclohexyl-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4S)-4-[4-(5-phenyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
N-[(2,5-difluorophenyl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl](pyridin-4-ylmethyl)amine
5-(azocan-1-yl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(4aS,8aS)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridine-2-carbonyl]benzonitrile
N-{5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl}acetamide
N-(2-hydroxyethyl)-1-{1-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
8-[(2,4,5-trimethoxyphenyl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(4-methoxy-2-methylphenyl)-3-(piperidin-1-yl)azetidine-1-carboxamide
5-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}imidazolidine-2,4-dione
(1s,4s)-4-[(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)methyl]cyclohexan-1-amine
1-(2-chloroprop-2-en-1-yl)-3-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
1-[(3-methoxyphenyl)methyl]-5-{methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}azepan-2-one
1-(6-phenylpyridazin-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2-methylpyridin-4-yl)-4-(3-methylthiophene-2-carbonyl)-1,4-diazepane
7-(2-methylphenyl)-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,7aR)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2,3-dihydro-1H-inden-2-amine
N-[3-(propan-2-yloxy)propyl]-3-(pyridin-4-yl)propanamide
4-({[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}methyl)-1-methylpiperidin-4-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-(1-benzoxepine-4-carbonyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,2S,9R)-11-{pyrazolo[1,5-a]pyridine-7-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-(4-methoxyphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
(4-{[3-(trifluoromethyl)phenyl]methyl}-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl)methanol
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
1-{1-[2-(2-methoxy-4-methylphenoxy)ethyl]piperidin-3-yl}pyrrolidin-2-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-methyl-4-[(5-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-1,2,4-oxadiazol-3-yl)methyl]piperidine
(3S,4R)-1-(1H-imidazol-4-ylmethyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
ethyl 4-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-amido}piperidine-1-carboxylate
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
N2-cyclopropyl-N4-[(2-methyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(methylsulfanyl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-methoxyethan-1-one
3-[4-(3-propoxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]pyridine
9-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-methylpropanamide
3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]naphthalen-2-ol
(3aR,5R,6S,7aS)-2-[(1-ethyl-1H-indol-4-yl)methyl]-octahydro-1H-isoindole-5,6-diol