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N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-(2-{[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]formamido}ethyl)piperidine-3-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1'-[1-(pyridin-2-yl)piperidine-3-carbonyl]spiro[indene-1,4'-piperidine]
1,4,6-trimethyl-2-oxo-5-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamido)-1,2-dihydropyridine-3-carboxamide
3-(azetidine-1-carbonyl)-N-[(2,6-dimethylpyridin-4-yl)methyl]benzene-1-sulfonamide
6-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[1-(4-methylphenyl)propyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
2-(3-{[(5-ethylpyrimidin-2-yl)(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
3-[5-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)thiophen-3-yl]prop-2-yn-1-ol
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(3-fluorophenoxy)ethan-1-one
5-(3-benzoylpiperidine-1-carbonyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-methyl-4-{1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
4-(cyclopentylsulfamoyl)-N-(2-oxopyrrolidin-3-yl)benzamide
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}[1-(4-methylpyridin-2-yl)propyl]amine
1-[(2,6-dimethoxyphenyl)methyl]-3-(3-methoxypropyl)piperidine
2-[4-(3-hydroxyphenyl)-6-methylpyrimidin-2-yl]phenol
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2H-1,3-benzodioxole-5-carboxamide
1,3-dimethyl-8-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}pyridine
3-phenyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,2,4-oxadiazole
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(trifluoromethyl)pyridin-2-yl]-decahydro-1,6-naphthyridin-2-one
N'1-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N'1-(2-methoxyethyl)cyclopropane-1,1-dicarboxamide
[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(3-methylphenyl)pyridine-3-carbonitrile
1-(2-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-(ethylamino)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)pyrimidine-5-carboxamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)morpholine
1-[(3-methylpyridin-2-yl)methyl]-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
(4aR,8aS)-1-[(3,4-dimethoxyphenyl)methyl]-6-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{1-[7-(2,5-dimethoxybenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-2-(dimethylamino)acetamide
(1S,5R)-6-[2-(4-fluorophenoxy)ethyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylpropanamide
3-amino-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-methyl-8-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethoxy}quinoline
N,1,3-trimethyl-2,6-dioxo-N-[1-(pyridin-3-yl)pentyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl 1-(2-hydroxy-3-{4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)piperidine-4-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]propanamide
2-(5-{[methyl(1-methylpiperidin-4-yl)amino]methyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]thiophen-3-amine
2-methyl-4-(4-{[3-(morpholine-4-carbonyl)piperidin-1-yl]methyl}phenyl)butan-2-ol
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)ethane-1-sulfonamide
3-cyclohexyl-1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)propan-1-one
2-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[2-methyl-4-(propylcarbamoyl)phenyl]piperidine-1-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]piperazin-2-one
7-fluoro-N,2-dimethyl-N-[(3-methyl-1H-indol-2-yl)methyl]quinoline-4-carboxamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
7-(oxolan-3-ylmethyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine