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N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}acetamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-(furan-3-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-phenyl-1H-imidazol-1-yl)acetamide
3-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
(3R,4S)-1-(isoquinolin-1-yl)-4-propylpyrrolidin-3-amine
6-butyl-2-{4-[(3-methylpiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
4-ethyl-1-[2-(ethylsulfanyl)ethyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1H-indol-1-ylmethyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[(1-cyclohexylpiperidin-3-yl)methyl][(2-fluoro-5-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1H-indazole-3-carboxamide
4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1-methylpiperidine
4-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-2-one
[3-(cyclopropylmethyl)-1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methanol
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
1-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-3-(3-fluorophenyl)propan-1-one
(2R,3R,6R)-5-cyclopentanecarbonyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,5-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3,7-dimethyl-1H-indol-2-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecane
7-(cyclohexylmethyl)-2-propanoyl-2,7-diazaspiro[4.5]decan-6-one
8-(oxane-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1-methyl-1H-pyrazole
N,6-dimethyl-2-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(2-methylphenyl)piperazine
5-{[2-(cyclohex-1-en-1-yl)ethyl](cyclopropylmethyl)carbamoyl}-1H-imidazole-4-carboxylic acid
1-[3-(3-methylphenoxy)azetidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(4aS,7aR)-N-ethyl-4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)acetamide
2-[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4-methyl-1H-imidazole
methyl 4-[({1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}formamido)methyl]benzoate
3-{4-[3-(3-chlorophenyl)-3-phenylpropanoyl]piperazin-1-yl}propanamide
7-methyl-3-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-(4-acetylphenyl)-3-[2-(propan-2-ylsulfanyl)ethyl]urea
3-cyclohexyl-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
N,2-dimethyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-1-phenyl-1H-1,3-benzodiazole-5-carboxamide
6-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-1,3-thiazole-4-carboxamide
4-cyclopropyl-6-[3-fluoro-5-(propan-2-yloxy)phenyl]pyrimidine
3-hydroxy-4-methoxy-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]benzamide
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-benzyl-3-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
(1R)-1-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2-phenylethan-1-amine
(3E)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylhex-3-enamide