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2-(furan-2-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}(methyl)({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-[2-(oxan-2-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
methyl 4-{[(3S,4R)-3-(3-methoxy-3-oxopropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}benzoate
2-methoxy-6-({3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(2R,3R,6R)-5-[(5-ethylpyridin-2-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-[1-(methoxymethyl)cyclobutanecarbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3E)-5,5-dimethyl-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}hex-3-enoic acid
4-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-2,3-dihydro-1,4-benzodioxine-6-carboxamide
14-[2-(benzylamino)pyrimidin-5-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanamide
2-{1-cyclopentyl-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(2-chloro-5-sulfamoylphenyl)-3-(propoxymethyl)pyrrolidine-1-carboxamide
(benzylsulfamoyl)(2-methoxyethyl)(thiophen-2-ylmethyl)amine
(1S,6R)-9-[1-(3,5-dimethylphenyl)piperidin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
3-(3-hydroxyquinoxalin-2-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]propan-1-one
1-[1-(propane-2-sulfonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-phenylpropanamide
ethyl 2-(4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholin-3-yl)acetate
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methoxyphenoxy)acetamide
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
2-(2-methyl-1,3-benzothiazole-6-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxyethyl)-1-[(1s,4s)-4-[(adamantan-2-yl)amino]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]acetamide
2-cyclopropyl-5-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
2-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-4H-3,1-benzoxazine-7-carboxamide
4-({2-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]-2H-1,3-benzodioxole-5-carboxamide
5-(1H-imidazol-1-ylmethyl)-2-{pyrazolo[1,5-a]pyridin-7-yl}pyridine
6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-(3-methylpentanoyl)-2,9-diazaspiro[5.5]undecan-3-one
[5-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[5-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
4-(1H-pyrazol-4-yl)-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]butan-1-one
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(4-methoxyphenyl)ethyl]propanamide
8-{[4-hydroxy-3-(prop-2-en-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-[2-(2,3-dimethoxyphenyl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine