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2-(2-chloro-6-methoxy-4-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)acetamide
4-{[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
4-(2,4-dioxoimidazolidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(1H-imidazol-1-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-butyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
4-(4-fluorophenyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1,2,3,6-tetrahydropyridine
2-[3-(2-cyclopentylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4H-chromen-4-one
N-(butan-2-yl)-N-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}cyclopentanamine
4-{1,3-dimethyl-4-[(3-phenylpiperidin-1-yl)methyl]-1H-pyrazol-5-yl}morpholine
2-(cyclopentylmethyl)-1-(3-methoxypropyl)-6-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-fluorophenyl)acetamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-(oxan-4-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[2-(propan-2-yloxy)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
3-(1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-2-yl)pyridine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-3-ethoxy-N-(1,3-thiazol-2-ylmethyl)propanamide
ethyl 1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxylate
(1S,5R)-6-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1-dimethyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
6-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine-1-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
1-(propan-2-yl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-[3-(4-fluorophenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclopentylacetamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-6-benzyl-3-(3-chloro-2-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl (1R,3S,3aR,6aS)-3-(5-acetylthiophen-3-yl)-1,5-diethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
1-(2,3-difluoro-4-methoxybenzoyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]pyrimidin-4-amine
2-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 4-{[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]amino}benzoate
N-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}methanesulfonamide
2-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]pyridine-4-carbonitrile
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-chloro-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
(4aS,8aR)-6-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-(6-methylpyridazin-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7,8-dimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
2-methanesulfonamido-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}acetamide
(2S)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-acetamidopropanamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
5-chloro-N-(3-hydroxy-2,2-dimethylpropyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide