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8-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
2-methyl-4-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyridine-3-carboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1-{2-[4-(hydroxymethyl)phenyl]acetyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{2-[4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazole
1-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(oxane-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethylpyrimidine-5-carboxamide
2-cyclooctyl-4-[4-(pyrazine-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[methyl(2-phenylethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
2-[2-(pyrimidin-2-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
(1S,6R)-9-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
3-[4-(9H-purin-6-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
2-({1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
1-{1-[2-(3-hydroxyphenyl)acetyl]piperidin-3-yl}-3-phenylpropan-1-one
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-1-(cyclohexylmethyl)-3-hydroxypiperidin-2-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
3-chloro-5-methoxy-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
3-ethyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidine-3-carboxylic acid
1-methyl-3-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-phenoxypyridin-3-yl)methyl]-1-(propan-2-yl)piperidin-4-amine
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
(3aR,7aS)-N-(1-cyclohexyl-1H-pyrazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
N-(3-methoxyphenyl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
(3S,4S)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
2,6-dimethyl-5-(2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
6-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoyl)-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
N-[3-(cyclopentyloxy)propyl]-8-fluoroquinoline-2-carboxamide
5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
4-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
N-butyl-3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(furan-2-ylmethyl)-2-methylpropanamide
2-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
2-(5-acetylthiophen-3-yl)-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]acetamide
4-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-2,7,8-trimethylquinoline
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-3-(4-methoxyphenyl)prop-2-enamide
N3-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}piperidine-1,3-dicarboxamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]piperidin-2-one
1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-N-[(3-methyloxetan-3-yl)methyl]piperidin-4-amine
(4aS,7aR)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-pentyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-{6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
(3R,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{4-[4-(3-cyanopyrazin-2-yl)piperazine-1-carbonyl]phenyl}cyclobutanecarboxamide