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[1-(2,3-dihydro-1H-indene-5-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
1-[2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)ethyl]piperidin-3-ol
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-(quinolin-8-yl)pyrrolidine-1-carboxamide
{2-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}urea
7-cyclopentyl-2-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1-(cyclopropanesulfonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[3-(4-methylpiperazin-1-yl)butyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-fluoro-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
[5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)furan-2-yl]methanol
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-4H-1,2,4-triazole
N-[3-(furan-2-amido)-4-methoxyphenyl]-4-methylpyridine-3-carboxamide
N-(3-ethoxy-2-hydroxypropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5-methyl-1,2-oxazole-3-carboxamide
2-phenyl-1-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)ethan-1-one
N-[(4-hydroxyazepan-4-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
9-(4-acetylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3-chlorophenyl)phenyl]-4-hydroxy-4-(hydroxymethyl)azepane-1-carboxamide
4-methyl-5-[4-(2-methylphenoxy)piperidine-1-carbonyl]pyrimidine
3-chloro-N-cyclopentyl-4-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]oxy}benzamide
4-(4-chlorophenyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}butanamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
6-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine
4-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-2-(trifluoromethyl)morpholine
1-(2H-1,3-benzodioxol-5-yl)-5-(5-ethyl-1,3-oxazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazole
5-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-[(3R,5S)-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrrolidin-3-yl]furan-2-carboxamide
(3S,4R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-methylpiperidine-3,4-diol
(2S)-2-acetamido-4-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]pentanamide
(3R,4S)-1-(4-methanesulfonylbenzoyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}acetic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
6-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-methyl-1H-indole-2-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide
2-(cyclopropanesulfonyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-cyclopropyl-3-{5-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(1-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]pyrrolidine-1-sulfonamide
5-(2-chlorophenyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]furan-2-carboxamide
(2S)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-acetamido-3-(1H-imidazol-4-yl)propanamide
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-({1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}oxy)pyridine
4-ethyl-3-({1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-8-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,5S)-1-benzyl-N-[2-(dimethylamino)ethyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-1-(oxolane-2-carbonyl)piperidin-4-amine