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N,N,2-trimethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-sulfonamide
N-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-imidazole-2-carboxamide
2-(2-hydroxyethyl)-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(cyclopropylmethyl)-1-(pyrrolidine-1-sulfonyl)piperidine-3-carboxylic acid
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(phenylsulfanyl)acetamide
8-(butan-2-yl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,3-diphenylpiperidine
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-4-yl)acetamide
3-{1-[2-(ethylsulfanyl)propanoyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2,6-dimethylphenol
3-(2,5-dimethoxyphenyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidine
(4aR,7aS)-1-benzyl-4-(2-hydroxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-ethyl-N4-methyl-N4-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidine-2,4-diamine
[3-(3-methoxypropyl)-1-(pyrimidin-5-ylmethyl)piperidin-3-yl]methanol
(1R,2S)-1-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-2,3-dihydro-1H-inden-2-ol
3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4-methylbenzene-1-sulfonamide
3-[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(prop-2-en-1-yl)amino]-1λ6-thiolane-1,1-dione
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(3-hydroxypropanoyl)pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
5,6-dimethyl-N-[1-(pyridin-4-yl)propan-2-yl]thieno[2,3-d]pyrimidin-4-amine
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-(3-chlorophenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
2-(adamantan-1-yl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
3-cyclopropyl-1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-{1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N,N-dimethylpyrrolidin-3-amine
1-(1'-{[3-(2-aminoethyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
N-{4-[4-(4-methoxypiperidin-1-yl)piperidin-1-yl]phenyl}-3-phenylpropanamide
N3-cyclohexyl-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
8-(1H-imidazol-2-ylmethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-chlorophenyl)-N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-(2,2-diethylcyclopropanecarbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-[(4-methylphenyl)methyl]-4-[6-(morpholin-4-yl)pyrimidin-4-yl]piperazin-2-one
3-{[3-cyclopentyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-1-methylimidazolidine-2,4-dione
N5-cycloheptyl-1-cyclopropyl-4-oxo-N3-(propan-2-yl)-N3-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(5-chlorothiophen-2-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{1-[1-(4-fluoro-3-methylbenzoyl)piperidin-4-yl]ethyl}morpholine
4-(2-methanesulfonylacetyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[4-(hydroxymethyl)phenyl]-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(1H-imidazol-4-yl)ethyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
4-[(2-hydroxyethyl)sulfanyl]-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]benzamide
5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-{2-[4-fluoro-3-(hydroxymethyl)phenyl]phenoxy}propanamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(3R)-4-hydroxy-3-methylbutyl]butanamide
N-{[1-(furan-2-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide