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1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
3-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methyl-2-oxopentanamide
1-(thian-4-yl)-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazine
2-amino-4-(3-hydroxyphenyl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
2-(5-acetylthiophen-3-yl)-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
1-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperidin-3-yl]pyrrolidin-2-one
N-(1H-imidazol-2-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
(butan-2-yl)({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})[(4-methylphenyl)methyl]amine
3-butyl-1-methyl-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
N-cyclohexyl-2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)butanamide
ethyl 2-chloro-5-({2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}amino)benzoate
3-(5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]propanamide
(1R,3S)-3-{[3-(2-fluorophenyl)propyl]carbamoyl}cyclopentane-1-carboxylic acid
N,N-diethyl-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine-3-carboxamide
1-[(3-chloro-1-benzothiophen-2-yl)methyl]-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
6-ethyl-4-{[3-(pyridin-3-ylmethyl)piperidin-1-yl]methyl}-2H-chromen-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-(pyrazin-2-yl)piperidin-3-yl]propanoic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[2-(methylsulfanyl)phenyl]methyl}piperazin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
4-[3-(1-methoxyethyl)phenyl]-N,6-dimethylpyrimidin-2-amine
N-[(4-hydroxyphenyl)methyl]-1-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(3-{[1-(ethanesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1,3-benzothiazole
2-({[(3R,4R)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetyl]azetidine-2-carboxylic acid
4-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)benzoic acid
7-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
9-(6-aminopyrimidin-4-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-8-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
5-fluoro-1-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1H-indole-2-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3,5-dimethyl-1,2-oxazole-4-sulfonamide
6-ethyl-N2,N2-dimethyl-N4-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrimidine-2,4-diamine
6-ethyl-2-[3-({[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3-[5-(6-oxo-1,6-dihydropyridin-3-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-(cyclohex-1-en-1-ylmethyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
9-ethyl-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{2-methyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}ethan-1-amine
(4aS,8aR)-6-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-methylpiperidin-3-amine
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(1-methyl-5-oxopyrrolidin-3-yl)urea
2-[({2-[4-(dimethylamino)phenyl]ethyl}amino)methyl]-6-fluoroquinolin-4-ol
N-[(2,3-dimethoxyphenyl)methyl]-3-[(2-fluorophenyl)formamido]propanamide
2-(furan-2-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-oxoacetamide
4-{5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine