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4-[3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]morpholine
2-{9-[(3-ethenylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-methyl-4-({4-methyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
2-(ethanesulfonyl)-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}[(2-methylphenyl)methyl]amino)ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-4-(trifluoromethyl)benzamide
3-hydroxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
5-chloro-3-methyl-2-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-indole
N4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methylpyrimidine-2,4-diamine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-(2-hydroxyethyl)-8-(4-oxo-4-phenylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[(propan-2-ylsulfanyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-benzyl-2-ethyl-N,6-dimethyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-(hydroxymethyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-ol
5-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]isoquinoline
3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
1-(4-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}phenyl)ethan-1-one
(2S,4R)-4-(2-cyanobenzamido)-N-ethyl-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
5-fluoro-3,8-dimethyl-2-(1H-pyrazol-3-yl)quinoline
4-[(dimethylamino)methyl]-1-(2,6-dimethylquinoline-4-carbonyl)azepan-4-ol
[9-(2-methoxyethyl)-3-(1H-pyrazole-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
5-(1-cyclopropyl-1H-pyrrol-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-ethyl-3-[1-(isoquinoline-5-carbonyl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(dimethylamino)-2-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
2-(4-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-1-yl)-1,3-benzoxazole
3-(benzyloxy)-1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidine
(3S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,5-dimethyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
6-amino-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}pyridine-3-carboxamide
1-methyl-N-(thiophen-3-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(3S,4S)-4-(dimethylamino)-1-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)pyrrolidin-3-ol
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(furan-2-yl)-5-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,4-triazole
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(1,2-oxazinan-2-yl)propan-1-one
(1R,5S,6R)-3-[3-(pyridin-3-yl)propanoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
(4aS,8aR)-6-[(4-methanesulfonylphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-(dimethyl-1,3-thiazol-5-yl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[1-(2-methylpropyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
N-ethyl-2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-4-fluoro-N,2-dimethylbenzamide
N-(1-benzothiophen-2-ylmethyl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
N-[4-(2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethoxy)phenyl]propanamide
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2-[methyl(piperidin-4-yl)amino]acetamide
2-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
N-(2H-1,3-benzodioxol-5-yl)-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-3-amine
7-(2-phenylethyl)-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-{[2-(2-aminoethyl)quinazolin-4-yl](methyl)amino}ethyl)piperidin-2-one