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3-(4-hydroxybutyl)-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
9-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3,9-diazaspiro[5.6]dodecane
4-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
N-[(3-fluoro-4-methylphenyl)methyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(3-chloro-2-fluorophenyl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
1-methyl-2-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
5-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-2-methoxyphenol
1-(4-fluoro-2-methylphenyl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1-(pyridin-2-ylmethyl)piperidin-4-amine
N-(2-phenylpropyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-(2-fluorophenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxylic acid
N-ethyl-5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
(2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-8-methylquinolin-3-yl)methanol
4-(2-fluoro-4-methylphenyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
N-(adamantan-2-ylmethyl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
(2S,3R)-2-amino-3-methoxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-[(1S,2S)-2-hydroxycyclohexyl]-N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
(3R,4S)-1-(2-propoxybenzoyl)-4-propylpyrrolidin-3-amine
2-[ethyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(6-methylpyridin-2-yl)methyl]pyridin-2-amine
2-[3'-oxo-1-(1H-pyrazole-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl]-N-(propan-2-yl)acetamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-{3-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
S-(2-cyclopentanecarbonyl-1,2,3,4-tetrahydroisoquinolin-6-yl)-3-hydroxybutane-1-sulfonamido
1-(4-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}thiophen-2-yl)ethan-1-one
5-(pyrimidin-5-yl)quinolin-8-ol
2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]benzoic acid
N-methyl-N-(oxolan-2-ylmethyl)-4-(propylsulfamoyl)benzamide
1'-[(3,4-dimethoxypyridin-2-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-(5-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
3-[(5-acetyl-4-methylpyrimidin-2-yl)amino]-N-cyclohexylpropanamide
3-(1-benzothiophen-7-yl)-4-methoxybenzamide
4-[5-(methoxymethyl)furan-2-carbonyl]-1,4-oxazepan-6-ol
3-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylpropanamide
3-methyl-1-(2-methylpropyl)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperazin-2-one
N-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]methanesulfonamide
7-(1-methylpiperidine-3-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-methyl-N-[4-(1H-pyrazol-3-yl)phenyl]propanamide
(2S,4S)-4-acetamido-N-ethyl-1-{[4-(furan-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-ol
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(naphthalen-2-yloxy)propanamide
1-(3-methylpiperidin-1-yl)-3-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}amino)propan-1-one
6-ethyl-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
benzyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(3-methylpyridin-2-yl)methyl]amine
2-(2,6-dimethylphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
4-(5-methylpyridin-2-yl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-ol