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8-[(5-methylfuran-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(furan-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
3-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(4aR,7aS)-1-(2-{[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
6-butyl-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,2-dimethyl-2-(morpholin-4-yl)propanamide
4-chloro-2-hydroxy-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]benzamide
3-hexyl-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-6-methoxypyrimidin-4-amine
2-(adamantan-1-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
(3R,4S)-4-cyclopropyl-1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
1-(cyclobutylmethyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(5-chloro-2-methoxyphenyl)-3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]propanamide
[(2S,6S)-4-[2-(3-fluorophenyl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-methyl-6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridazine
2-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-6-methoxyphenol
4-methoxy-N-(2-methoxyethyl)-2-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-5-phenyl-1H-pyrazole-3-carboxamide
N-(furan-3-ylmethyl)-N-[(3-methylthiophen-2-yl)methyl]cyclopropanamine
3-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methoxy-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}benzoic acid
(1R,3S)-3-methoxy-7-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-{5-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[4-({5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-N'-(4-methylphenyl)propanediamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-methoxypropan-1-one
7-(3-chlorophenyl)-4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(3S,4S)-1-(2-propylpyridine-4-carbonyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-{2-[(1-ethenyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2-methylpropan-1-one
1-cyclopentyl-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-oxopyrrolidine-3-carboxamide
3-(3-methylphenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
5-ethyl-N,2,3-trimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
5-(2-fluorophenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-(2-hydroxy-5-methylbenzoyl)-3-propylpiperidine-3-carboxylic acid
(2S,4S)-4-(cycloheptylamino)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
8-[2-(2-hydroxyethoxy)ethyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(1S,6R)-9-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(2-methyl-5-sulfamoylphenyl)urea
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
(3R,4S)-1-(3-methoxy-4-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-amine
2-methyl-7-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-{2-methyl-4-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenoxy}acetamide
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide
2-[4-(2-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide