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3-[2-(2,6-difluorophenyl)ethyl]-1-(1,3-thiazol-2-yl)piperidine
5-propyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
8-(5-methoxypyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3-ethoxypropyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
2-({2-[(2,2-dimethyloxan-4-yl)(ethyl)carbamoyl]phenyl}amino)acetic acid
2-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
methyl({[4-(1H-pyrazol-5-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
3-[6-amino-5-cyano-4-(6-methyl-2H-1,3-benzodioxol-5-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}pyrazolo[1,5-a]pyridine-2-carboxamide
methyl 4-{[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]methyl}benzoate
(2R)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]oxolane-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
6-(benzyloxy)-4-cyclopentyl-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
1-cyclohexyl-3-hydroxy-4-[2-(propan-2-yl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(cyclohexylmethyl)-1,4-diazepan-5-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
2-(4-fluorophenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
4-(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazine-2-carbonyl)morpholine
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methoxypropan-1-one
N-(4-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)acetamide
5-methyl-3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-methoxypiperidine-1-carboxamide
N-[(1R,3S)-3-(morpholine-4-carbonyl)cyclopentyl]-3-phenyl-1,2-oxazole-4-carboxamide
(2R,6S)-4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2,6-dimethylmorpholine
1-[4-(3-hydroxyphenyl)piperidin-1-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-(2-methoxyethyl)-4-methyl-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
3-cyclopropyl-6-[1-(4-methoxyphenyl)cyclopropyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-methoxy-5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}benzoic acid
3-cyclopropyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
1-(1-benzylpiperidin-4-yl)piperidine-3-carboxylic acid
4-[1-(1-benzylpyrrolidin-3-yl)-1H-imidazol-2-yl]-3-methoxyphenol
2-[3-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]-2,3-dihydro-1H-isoindol-1-one
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-phenoxy-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butan-1-one
N-(2,4-dimethoxyphenyl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
(4aS,7aR)-1-[(2-ethoxyphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-hydroxypropyl)-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclobutylmethyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-3-{5-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
6-chloro-2-[4-(pyrimidin-4-yl)-1,4-diazepan-1-yl]-1,3-benzothiazole
5-amino-3-(4-fluoro-3-methoxyphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
(3R,5S)-N-butyl-5-[(4-methylpiperazin-1-yl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperazine
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
N-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
1-[(4aS,8aS)-4a-hydroxy-7-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
2-(5-{[(2-ethyl-6-methylpyridin-3-yl)oxy]methyl}-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl)acetamide