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4-(1-benzothiophen-2-ylmethyl)-11-[(1,2-oxazol-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(N-benzyl-1-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidin-5-yl}formamido)propanamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
methyl (2R)-2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-(methylsulfanyl)propanoate
2-amino-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-6-(propan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,4R)-1-(4-chlorobenzoyl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
N-[2-(5-methylfuran-2-yl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
1-(2-methoxy-6-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]pyridine-3-carbonitrile
[2-(diethylamino)-2-(furan-2-yl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
[(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-benzoyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]piperidin-4-amine
4-{3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N-[(6-{4-[(4-hydroxy-3-methylphenyl)methyl]piperazin-1-yl}pyridin-3-yl)methyl]acetamide
6-(2-hydroxyethyl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(furan-3-ylmethyl)(methyl)(quinolin-4-ylmethyl)amine
1-{[3-(2-methylphenyl)phenyl]methyl}-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
N-methyl-N-(quinolin-5-ylmethyl)-4-(1H-1,2,4-triazol-3-yl)benzamide
methyl 1-ethoxy-8-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
9-ethyl-N-(3-fluorophenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-hydroxy-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
3-benzyl-1-methyl-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-2,3-dihydro-1H-indol-2-one
2-hydroxy-5-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)benzoic acid
N-(3-chloro-4-methoxyphenyl)-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
5-({[2-(2,3-dihydro-1H-indol-1-yl)ethyl]carbamoyl}amino)-2-methoxy-N,N-dimethylbenzamide
4-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
1,3,6-trimethyl-N-[2-methyl-1-(pyridin-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]amino}ethan-1-one
N-(3-chloro-4-propanamidophenyl)-4-acetamidobutanamide
[1-(2-chloro-5-fluorobenzoyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-[3-(1H-imidazol-1-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-({2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
N'-(2-chlorophenyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)ethanediamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
2-[4-carboxy-4-(cyclopropylmethyl)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperidin-4-ol
(4aS,8aR)-1-butyl-6-[5-(methoxymethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[4-(4-hydroxyphenyl)butan-2-yl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-2-{[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
2-(carbamoylamino)-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]acetamide
4-{[(2-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(1,3-thiazol-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
2-(3-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
N-methyl-N-({4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)methanesulfonamide
3-(5-tert-butyl-2-methoxyphenyl)-1-methyl-1-[4-(morpholin-4-yl)butyl]urea
2-{5-[(2,4-difluorophenyl)methyl]-1,2,4-oxadiazol-3-yl}pyrimidine