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3-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
N-ethyl-2-{4-[6-(3-fluorophenyl)pyridine-3-carbonyl]piperazin-1-yl}acetamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-{4-[(2,4-difluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-6-fluoro-N,3-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
ethyl 4-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-3-yl]piperazine-1-carboxylate
1-(benzenesulfonyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
2-(4-fluorophenyl)-2-hydroxy-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxypropyl)-N-methylacetamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(2-hydroxyethyl)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-(pyrrolidin-1-yl)butan-1-one
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-methylpiperazin-2-one
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(3-fluoro-4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4,6-dimethyl-3-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-1,2-dihydropyridin-2-one
3-(cyclobutylsulfamoyl)-N-[3-(pyridin-2-yl)propyl]benzamide
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(4-phenoxyphenyl)methyl]amine
3-({4-[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-1H-indole
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
2-{8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methylthiophen-2-yl)methyl]benzamide
2-cyclohexyl-5-{1-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-imidazol-2-yl}pyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}morpholine
[(5-chlorofuran-2-yl)methyl][(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
(4aR,8aR)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-2H-1,4-benzoxazine
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-6-(methoxymethyl)pyrimidine
6-(4-fluorophenyl)-N-[(2S)-1-hydroxybutan-2-yl]-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[2-(3,5-dimethylphenoxy)ethyl]-N-methylacetamide
1-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
5-[1-(3,3-dimethylbutyl)pyrrolidin-2-yl]-N-[2-(pyrazin-2-yl)ethyl]thiophene-2-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(pyridin-2-yl)propyl]-6-{[1-(pyridin-3-yl)ethyl]amino}pyridine-3-carboxamide
3-methoxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
1-[2-methoxy-5-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-ethyl-8-[(8-methoxyquinolin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1,3-dihydroxy-2-methylpropan-2-yl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methoxypropanamide
6-amino-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]pyridine-2-carboxamide
8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(2S,4S)-N-ethyl-4-[2-(2-methylphenyl)acetamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(piperidin-1-yl)ethyl]acetamide
N-(1-methoxybutan-2-yl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
1-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}methyl)-N,N-dimethylcyclohexan-1-amine