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2-[methyl(pyridin-4-ylmethyl)amino]-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
2-({[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
1-(4-{[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}piperidin-1-yl)ethan-1-one
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(oxolane-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-N,N-dimethyl-3-[2-(morpholin-4-ylmethyl)phenyl]-1H-1,2,4-triazol-5-amine
(3R,4R)-1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
5-butyl-1'-(5-methylpyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{2-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}piperazin-2-one
N4-[2-(diethylamino)ethyl]-N4-methyl-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-methoxy-3-{[4-(pyrrolidin-3-yl)piperazine-1-carbonyl]amino}benzoate
(2R,6R)-4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
methyl 8-(furan-3-ylmethyl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[4-(pyridin-2-yl)butyl]-2-(pyrrolidin-3-yl)benzamide
(2R,6S)-4-[6-(3-chlorophenyl)-3-(piperidine-1-carbonyl)pyridin-2-yl]-2,6-dimethylmorpholine
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(1H-imidazol-2-yl)piperidine
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrazole-4-carboxylate
6-cyclopentyl-1-methyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-(pyridin-4-yl)propanamide
2-[1-(2-phenylethyl)-4-(1-phenylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
N-[2-(4-fluorophenyl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
1-{3-methyl-5-[2-(1,1,2,2-tetrafluoroethoxy)phenyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-phenyl-1,4-diazepane
(5S)-5-(3-oxo-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propyl)imidazolidine-2,4-dione
N-cyclobutyl-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
(2R)-2-[(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propanamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(5-methylfuran-2-yl)methyl]acetamide
methyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-[2-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
2-(dimethylamino)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(4-fluorophenyl)acetamide
1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-2-ol
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
3-(cyclopropylmethyl)-1-(2,3-difluoro-4-methoxybenzoyl)piperidine-3-carboxylic acid
2-ethyl-N-[(5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl)methyl]butanamide
2-methyl-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-1,3-benzothiazole-6-sulfonamide
ethyl 4-[(2-chlorophenyl)methyl]-1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxylate
2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
4-{4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[5-(morpholine-4-carbonyl)furan-2-yl]isoquinoline
N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide