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3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(oxane-4-carbonyl)piperidine
3-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pentan-3-amine
4-(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)morpholine
3-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydroquinolin-2-one
(2S,4R)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-[2-(morpholin-4-yl)acetamido]pyrrolidine-2-carboxamide
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
2-benzyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1,3-thiazole-4-carboxamide
1-[(4aR,8aS)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
N-cyclopropyl-4-methoxy-2-({1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}oxy)benzamide
N-butyl-9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-4-chloro-1H-pyrrole-2-carboxamide
5-[4-(4-methyl-1H-imidazole-5-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
4-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)piperidin-4-amine
3-(hydroxymethyl)-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
4-{4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-(3-methylbutyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[4-(morpholin-4-yl)butyl]-4-phenylpiperidin-4-ol
9-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(4-chloro-1H-pyrazol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
{1-[1-(2-methyloxane-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
4-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)benzamide
(3S,4R)-3-ethyl-1-[3-(2-methoxyphenyl)benzoyl]-4-methylpiperidin-4-ol
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-4-[(2-methylpropanamido)methyl]benzamide
N-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-[(1S,5R)-3-[(2-cyanophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(2S,4R)-N,N-diethyl-1-(4-ethylbenzoyl)-4-propanamidopyrrolidine-2-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2,4-dimethylpyrimidine-5-carboxamide
8-(3-methoxypropyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-amino-2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
2-methyl-N-{2-[methyl(pyridin-2-ylmethyl)carbamoyl]phenyl}furan-3-carboxamide
3-(2-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one
4-(1H-imidazol-1-ylmethyl)-1-[3-(piperidin-4-ylmethyl)benzoyl]piperidin-4-ol
2-(2-methylpropyl)-8-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]sulfonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-methyl-3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}urea
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]-1-ethyl-1,2-dihydropyridin-2-one
(2S)-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
2-acetamido-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
1-(6-methyl-3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
6-benzoyl-1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(2-methylpropyl)amine
2-[3-(3,4-difluorophenyl)-5-[1-hydroxy-3-(methylsulfanyl)propyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
(1s,4s)-4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]cyclohexan-1-ol
{3-[(2-fluorophenyl)methyl]-1-(9H-purin-6-yl)piperidin-3-yl}methanol