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N-[(5-ethylpyridin-2-yl)methyl]-6-methoxy-N-methylpyrimidin-4-amine
3-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2-(1H-indazol-3-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-6-methoxyphenol
6-methyl-2-oxo-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(pentan-3-yl)({2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl})amine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[(1-methyl-1H-pyrazol-3-yl)carbamoyl]methyl}-decahydro-2,7-naphthyridine-2-carboxamide
2-[2-(propan-2-yl)-1,3-thiazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(1,3-thiazol-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-benzyl-N,N-dimethyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(dimethylamino)-3-{2-[(4-methanesulfonylpiperazin-1-yl)methyl]-4-methoxyphenoxy}propan-2-ol
1-[(4aR,8aS)-1-(4-tert-butylbenzoyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
5-[3-(1-benzyl-1H-pyrazol-3-yl)phenyl]pyrimidine
methyl 1-ethoxy-8-[2-(methylsulfanyl)pyridine-3-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(4-chloro-2-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenoxy)acetic acid
2-{4-[(4-aminopiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
8-(2-methoxybutanoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(cyclopent-2-en-1-yl)ethan-1-one
9-[(2-fluoro-5-methoxyphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-5-(7-methyl-1H-indol-3-yl)thiophene-2-carboxamide
3-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
1-(1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indol-3-yl)butan-1-one
1-(5-methoxypyridin-3-yl)-1H-1,3-benzodiazole
3-[4-(furan-2-yl)butan-2-yl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-[cyclopropyl(pyridin-2-yl)methyl]-5-methoxy-N,1,2-trimethyl-1H-indole-3-carboxamide
6-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}pyridine-3-carbonitrile
3,3-dimethyl-1-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}urea
4-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-4-[(2,3-difluorophenyl)methyl]piperazin-2-one
2-amino-6-(2,2-dimethyloxan-4-yl)-5-methyl-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
4-{4-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]phenyl}but-3-yn-1-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(4-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[(2,3-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[3-(4-chlorophenyl)piperidin-1-yl]methyl}benzoic acid
5-methoxy-2-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}phenol
(1H-1,3-benzodiazol-2-ylmethyl)[(2-methoxyphenyl)methyl]propylamine
3-(6-methoxypyridin-3-yl)-1-[2-(3-phenylpiperidin-1-yl)ethyl]urea
2-methyl-N-[3-(2-propoxyphenyl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-cyclopropyl-4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)benzamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-phenyl-1H-pyrazole-5-carboxamide
5-ethyl-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]thiophene-2-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1-methylpyrrolidin-2-yl)acetamide
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-benzyl-N-(2-hydroxyethyl)piperidine-4-carboxamide
N-ethyl-2-{4-[3-(furan-2-yl)-3-phenylpropanoyl]piperazin-1-yl}acetamide
1-{1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}-N,N-diethylpiperidine-3-carboxamide
6-(6-methoxypyridin-3-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
6-methyl-3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one