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(2E)-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-4-yl)prop-2-enamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-[(2-methylpyrrolidin-1-yl)sulfonyl]benzamide
[(1-cyclopentylpiperidin-4-yl)methyl][(3-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
(4aS,7aR)-1-[(6,8-dimethyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
5-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
dimethyl({4-methyl-5-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(3-methylbenzoyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-8-(trifluoromethyl)quinolin-4-amine
(4aS,7aR)-1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
3-methyl-1-[2-(phenylsulfanyl)ethyl]-1,2-dihydroquinoxalin-2-one
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzothiazol-2-amine
7-[(5-methoxy-1H-indazol-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-(2H-1,3-benzodioxol-5-yl)-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}benzamide
[(3R,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(2,3-dihydro-1H-inden-2-yl)-2-ethyl-4-methyl-N-propyl-1,3-oxazole-5-carboxamide
N-[(3R,4S)-4-(propan-2-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanesulfonamide
1-methyl-4-phenyl-3-[1-(2-phenylethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2-chloro-4-fluorophenoxymethyl)-N-(2,3-dihydro-1H-inden-2-yl)-1,2-oxazole-3-carboxamide
8-[2-(dimethylamino)benzoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(quinolin-3-yl)phenoxy]acetic acid
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(5-methylthiophene-3-carbonyl)-6-(morpholin-4-yl)-decahydroisoquinoline
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylpropyl)piperidine
N-[(3S,5S)-1-(cyclopentylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-ethylpyrimidine-5-carboxamide
(2R,6R)-4-[2-(dimethylamino)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
4-[(5-cyclopentylthiophen-2-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
N-(3,4-dimethylphenyl)-4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carboxamide
(3R)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6-dimethylpyridine
N-(4-{4-[(2,3-dihydroxypropyl)(methyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
4-(2-fluorophenoxy)-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxylic acid
N-[(2R)-3-methylbutan-2-yl]-2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
4-methoxy-3-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)carbamoyl]amino}-N-methylbenzamide
2-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-1,2-oxazolidine
N-methyl-3-({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}sulfamoyl)-N-propylbenzamide
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepane-6-carboxylic acid
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4-{[2-(dimethylamino)-1-phenylethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-[(4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]pyridin-2-amine
N-{2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
2-{3-[3-(3-cyano-6-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-N,N-dimethylacetamide
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide