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N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-{[(2-fluorophenyl)methyl](methyl)amino}acetamide
5-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
3-methyl-2-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-(thiophen-3-ylmethyl)piperidine
methyl (2R,4S)-4-hydroxy-1-(naphthalene-2-sulfonyl)piperidine-2-carboxylate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-methyl-6-(4-{[3-(methylsulfanyl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
1-(1,4-dioxan-2-ylmethyl)-5-(methoxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
1-(cyclohexyloxy)-3-{[1-(pyrimidin-2-yl)piperidin-4-yl]amino}propan-2-ol
1-{3-[3-(3-fluorophenoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(3S)-2-oxoazepan-3-yl]acetamide
6-chloro-2-methyl-4-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
N-butyl-N-(furan-2-ylmethyl)-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-(pyridin-2-ylsulfanyl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
methyl 3-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
3,3-dimethyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
N-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}phenoxy)acetic acid
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
(2E)-3-(1H-imidazol-4-yl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}prop-2-en-1-one
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
6-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]pyrazine-2-carboxamide
4-{[1-(methoxymethyl)cyclopentyl]sulfamoyl}-N-propylbenzamide
7-fluoro-4-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
(3R)-3,4,4-trimethyl-1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-3-ol
5-[4-(3-methylpiperidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
(2S)-N-ethyl-1-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
3-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)-N-(2-ethylphenyl)propanamide
1-[5-(5-ethyl-1,2-oxazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]-4-methylpiperazine
N-[(3S)-1-benzylpyrrolidin-3-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-fluoro-N-{1-[1-(3-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(2,6-dimethylpyridin-4-yl)-4-[3-(1H-imidazol-2-yl)benzoyl]piperazine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-{4-[3-(methoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl}pyridine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-1,3-thiazole-5-carboxamide
9-[3-(ethylsulfanyl)propanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2,6-diamino-4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
[3-({1-[(2,3,5-trifluorophenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
N-methyl-N-{2-[1-(2-methylpyridin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
5-(cyclohexylamino)-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-{[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}acetamide