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4-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyridine-4-carbonyl}morpholine
N6-benzyl-N5-methyl-N5-(1,3-thiazol-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]piperidin-4-ol
2-(methylsulfanyl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
1-(4-fluorophenyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepane
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopropane-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(methylsulfanyl)butyl]piperazine
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-ethylpiperidin-3-ol
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-ethyl-2-(4-methyl-1,4-diazepan-1-yl)-N-(2-methylprop-2-en-1-yl)acetamide
N-[(3S,4R)-1-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)-4-propylpyrrolidin-3-yl]acetamide
methyl 5-{2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
1,9-dimethyl-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}oxane-4-carboxamide
2,3-dimethyl-7-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2S)-3-phenyl-2-{[4-(piperidin-1-ylmethyl)phenyl]formamido}propanamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-amine
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
1-(3-hydroxypropanoyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
4-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methylbenzamide
N-[(2-methoxypyrimidin-5-yl)methyl]-4-(2-methyl-1H-imidazol-1-yl)aniline
1-[(3-ethenylphenyl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
2-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 5-[(3-methylbutyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
1-(5-{[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
1-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(2S,4S)-N,N-diethyl-4-[2-(4-fluorophenoxy)acetamido]-1-methylpyrrolidine-2-carboxamide
2-hydroxy-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-3-(2-methylphenoxy)propan-1-one
2-methyl-4-[2-(propan-2-yloxy)phenyl]-1H-imidazole
N-cyclobutyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(3-chlorophenyl)-4-[6-(propan-2-yl)pyridazin-3-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-5-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-chloro-5-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
6-methyl-5-{5-[5-(3-methylphenyl)furan-2-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
ethyl 1-(3-{[(1-hydroxycyclohexyl)methyl]carbamoyl}-6-(4-methylthiophen-2-yl)pyridin-2-yl)piperidine-4-carboxylate
7-[2-(furan-2-yl)azepane-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
4-(1H-imidazol-2-yl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine
2-{2-methylthieno[2,3-d]pyrimidin-4-yl}benzoic acid
methyl 5-[(2-methylbutyl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(naphthalen-2-yl)acetamide
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-ethyl-5-(5-propylfuran-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
{[5-(furan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
4-methoxy-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
N-ethyl-6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-methylpyrimidin-4-amine