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5-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[2-(dimethylamino)ethyl]piperazin-1-yl}-2-(4-phenoxyphenyl)acetic acid
4-(6-{pyrazolo[1,5-a]pyridin-7-yl}pyrazine-2-carbonyl)morpholine
2-(morpholin-2-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethan-1-one
(1S,6R)-9-(3-phenoxybenzoyl)-3,9-diazabicyclo[4.2.1]nonane
[(3R,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-methoxy-5-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
methyl 2-[8-(1,3-benzothiazol-2-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[(2-methylphenyl)methyl]-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}acetamide
(8aS)-2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
8-(3-aminophenyl)-2-methylquinolin-4-ol
N-(2-propoxyethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{1-oxaspiro[4.5]decan-3-yl}acetamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(1-methylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
dimethyl(3-{2-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N,N-dimethyl-3-[2-(morpholin-4-ylmethyl)phenyl]-1H-1,2,4-triazol-5-amine
N-{2-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenoxy]ethyl}acetamide
1-methyl-3-(propan-2-yl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-fluorophenyl)-4-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}piperazine
[(3R,5R)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-(3-chloro-4-methoxyphenyl)-3-[1-(cyclopropanesulfonyl)piperidin-3-yl]propanamide
2-(morpholin-4-yl)-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
5-methanesulfonyl-2-methyl-4-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)pyrimidine
(1R,9aR)-1-({[(1-methyl-5-phenyl-1H-pyrazol-3-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
6-oxo-N-(thiophen-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-fluoro-N-(furan-2-ylmethyl)-N-propylpyridine-4-carboxamide
2-amino-4-(1,2-dimethyl-1H-imidazol-5-yl)-5-methyl-6-phenylpyridine-3-carbonitrile
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-(2-methoxyethyl)-1-{1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
(2R,3R)-3-{[(3-hydroxy-4-methoxyphenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2-methylphenyl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
4-(2-ethyl-1-benzofuran-3-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
8-[2-(propan-2-yl)pyrimidine-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
5-chloro-6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid
6-[2-(2-chlorophenyl)-2-hydroxyethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{1-[1-(3-chloro-4-methylbenzoyl)piperidin-4-yl]ethyl}morpholine
2-(5-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}furan-2-yl)benzonitrile
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
1-[(3S,4R)-1-[1-(2-fluorophenyl)piperidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-(oxolan-2-ylmethyl)-N-propyl-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-amino-N-methyl-4-phenyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-sulfonamide
N-[(4-methoxypyridin-2-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
ethyl 1-(1-benzothiophen-2-ylmethyl)-3-(2-methoxyethyl)piperidine-3-carboxylate
3-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
2-methyl-1-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)azetidin-3-yl]piperidine
(2S)-2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}propanamide