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N-[(2-ethoxyphenyl)methyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
methyl[2-methyl-2-(morpholin-4-yl)propyl](4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-fluoro-1,2-dihydroquinolin-2-one
(3aS,6aS)-2-[(1-ethyl-1H-indol-5-yl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-4-ol
N-(1,4-dioxan-2-ylmethyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N,5-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-ethyl-N-{2-[methyl(phenyl)amino]ethyl}-5-oxopyrrolidine-3-carboxamide
methyl 3-[(adamantan-1-ylformamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
1-benzyl-N,N-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
2-{4-[3-(5-chloro-2-hydroxyphenyl)-1H-pyrazol-1-yl]phenyl}acetic acid
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2,2-diethylmorpholine
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-[methyl(2-phenylethyl)amino]-N-[2-(methylamino)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)acetamide
(3S,4S)-1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(dimethylamino)methyl]piperidin-3-ol
(2R,6R)-1-(1H-imidazol-2-ylmethyl)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-[4-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
3-butyl-1-methyl-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
4-methyl-6-[4-(2-propoxyethyl)piperazin-1-yl]-2-(pyridin-3-yl)pyrimidine
N-cyclopropyl-4-methoxy-3-({1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
2-(5-{1-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
N-[(3,5-difluorophenyl)methyl]-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3,6-dimethyl-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-amine
1-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[(4-hydroxypiperidin-1-yl)methyl]-N-(1-propylcyclopropyl)-1,2-oxazole-3-carboxamide
1-(benzenesulfonyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}cyclopropane-1-carboxamide
4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-amine
4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)thiomorpholine
1-{1-[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)phenyl]ethyl}piperidine
3-(2-methoxyethyl)-5-(thiophen-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
[(8-fluoroquinolin-2-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(3-fluorophenyl)methyl]morpholine
1-{1-[(3-methoxyphenyl)methyl]-5-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-3-(4-chloro-1H-pyrazol-1-yl)propanamide
2-{4-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}propanamide
{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
N-(cyclopropylmethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
2-ethyl-4-(1H-indol-2-ylmethyl)-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine