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3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,1-benzoxazole
(2R,3S,6R)-3-(4-methylphenyl)-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(2E)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-3-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
3-[(2,4-difluorophenyl)methyl]-1-(pyrazin-2-yl)piperidine-3-carboxylic acid
5-chloro-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)(oxan-4-ylmethyl)amine
N-benzyl-N-[(6-methylpyridin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{2-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]pyrimidin-4-yl}piperidin-4-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(5-hydroxypentyl)-5-methylpiperidin-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1-methyl-1H-indol-3-yl)acetamide
2-[(4-ethylphenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-ethyl-N-[2-(morpholin-4-yl)ethyl]quinoxaline-5-carboxamide
4-{4-[(3,4-difluorophenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-4-[3-(propan-2-yl)-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]pyridine
2-[3-(methoxymethyl)phenyl]-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]acetic acid
4-(4-{[4-(dimethylamino)azepan-1-yl]methyl}phenyl)-2-methylbutan-2-ol
N-({2-[4-fluoro-3-(hydroxymethyl)phenyl]phenyl}methyl)propanamide
5-(4-methoxyphenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(2-fluorophenyl)methyl]-2-{[1-(4-methanesulfonylphenyl)ethyl]amino}acetamide
({3-[(dimethylamino)methyl]-4-methoxyphenyl}methyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
2-[4-(3-acetyl-2-fluorophenyl)phenyl]-N,N-dimethylacetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)acetamide
1-tert-butyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-pyrrole-3-carboxamide
2-{4-[2-(2,3-dimethylphenoxy)ethyl]phenyl}acetamide
3-{6-[(3-methoxyphenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepane-1-carbonyl}pyridin-1-ium-1-olate
N-butyl-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(furan-2-ylmethyl)acetamide
N-(4-{[4-(5-{[(2-methylphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]methyl}phenyl)acetamide
(3R,4R)-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
3,3-dimethyl-1-{[5-(3-methylpyrazin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]amine
3-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}pyridine
N,N-dimethyl-2-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethane-1-sulfonamide
1-(3-cyclopentylpropyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-{[(2S,4S)-4-fluoro-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
7-(2-cyclohexylethyl)-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
methyl 1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
2-(4-tert-butylphenoxymethyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
(1S,5R)-6-benzyl-3-(2-methoxyacetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
({6,7-dimethoxy-2-[(4-methylphenyl)methoxy]quinolin-3-yl}methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
ethyl 3-({5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazol-3-yl}formamido)-5-methylhexanoate
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-ethoxyphenyl)methyl]pyrrolidine-2-carboxylate
1-{1'-[(3-hydroxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one