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2-[3-({[(3-methylphenyl)methyl](oxolan-2-ylmethyl)carbamoyl}amino)phenyl]acetamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridazine-4-carboxamide
6-[(oxan-4-yl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(1H-pyrazol-1-yl)benzamide
N-[(1-methylpiperidin-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
methyl({[5-(oxan-2-yl)furan-2-yl]methyl}){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-ethyl-3-(2,3,4-trimethoxyphenyl)benzamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-1-{4-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]piperidin-1-yl}propan-1-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
2-cyclopropyl-1-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,3-benzodiazole
2-[2-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)phenoxy]ethan-1-ol
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-{5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-yl}morpholine
5-(2-fluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,2,4-triazin-3-amine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide
2-amino-6-cyclopropyl-4-(2,3-dimethoxyphenyl)pyridine-3-carbonitrile
6-methyl-1-{3-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-(furan-3-ylmethyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
3-({3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}sulfonyl)pyridine
N-butyl-2-[(dimethylamino)methyl]-N-(thiophen-3-ylmethyl)-1,3-thiazole-4-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(2E)-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-3-yl)prop-2-enamide
3-methyl-8-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-methyl-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}thian-4-amine
3-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
1-(4-fluorophenyl)-4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}piperazine
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]benzamide
(2S)-2-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
(4aS,8aR)-1-(2-aminoethyl)-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
[5-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)furan-2-yl]methanol
N-[(2,5-dimethylphenyl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
9-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-methyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
1-[(1-benzyl-1H-imidazol-5-yl)methyl]piperidin-2-one
2-(4,6-dimethoxypyrimidin-2-yl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(oxolan-2-ylmethyl)acetamide
1-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N3-benzyl-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
2-(carbamoylamino)-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
2,3,6-trimethyl-N-{3-[(pyridin-3-yl)amino]propyl}quinoline-4-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide