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4-(1-ethyl-1H-imidazol-2-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
5-(4-{2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-[4-(1-benzofuran-2-ylmethyl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
(3R,4R)-4-amino-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-(2-methylphenyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
1-[(3-fluorophenyl)methyl]-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopentyl-3-(2-oxoimidazolidin-1-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
(4aR,8aR)-4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-octahydro-2H-1,4-benzoxazine
1-[2-(dimethylamino)ethyl]-N-methyl-6-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
3-methyl-7-{3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(3-chlorophenyl)-1-ethyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
2-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-6-methylpyridine
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-methyl-1H-indole
(2E)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}prop-2-enamide
{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
5-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-[(4-chlorophenyl)methyl]-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[1-(2,2-dimethylpropyl)piperidin-4-yl]methyl}-2-methoxy-2-methylpropanamide
1-(2H-1,3-benzodioxol-5-yl)-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]piperidine
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-(pyridin-3-yloxy)acetamide
N-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}methanesulfonamide
(4aS,7aR)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-3-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,2-oxazole-4-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
3-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
4-[4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]quinazoline
5,6-dimethyl-2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
6-(2-aminoethyl)-2-[3-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N,N-dimethyl-4-[3-(4-methylpiperazin-1-yl)pyrrolidine-1-carbonyl]aniline
6-ethoxy-3-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-ethyl-3-[2-(methylsulfanyl)ethyl]-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
(2S,4S)-N-ethyl-4-{4-[4-(morpholin-4-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(3-methanesulfonamidophenyl)urea
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
N-(2,3-dimethylquinoxalin-6-yl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-[2-(ethoxymethyl)-7-(oxan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(ethylamino)-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(morpholin-2-yl)ethan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-hydroxy-2-(4-methylphenyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(2-hydroxyethyl)-2-phenylacetamide
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carbonitrile
3-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-[(3-methoxyphenyl)methyl]-N-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-amine
4-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-4H-1,2,4-triazole
3-[5-(difluoromethyl)-1,2,4-oxadiazol-3-yl]-2-phenoxypyridine