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N-(2,3-dihydro-1H-inden-5-yl)-4-(pyrimidin-4-yl)piperidine-1-carboxamide
[(3R,4R)-1-(2-chloro-3-methylbenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-(2-{[4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-yl]amino}ethyl)piperidin-4-ol
4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-2-(4-methylpentyl)morpholine
3-hydroxy-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-oxo-N-(4-phenoxyphenyl)-2,8-diazaspiro[4.5]decane-8-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(3-methoxyphenoxy)azetidin-1-yl]propan-1-one
3-{[1-(1,4-dioxane-2-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dimethyl-N-(propan-2-yl)quinoxaline-6-carboxamide
1-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
2-methoxy-4-[(1E)-3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}prop-1-en-1-yl]phenol
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
6-methyl-2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
5-methyl-N-{3-[methyl(phenyl)amino]propyl}-1,3,4-oxadiazol-2-amine
2-({2-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-fluorophenyl)propan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(3-methoxyphenyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
(2S)-4-methyl-2-phenyl-1-[(5-propylfuran-2-yl)methyl]piperazine
N-[(5-phenylfuran-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-ethyl-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(2-methylphenyl)propanamide
9-cyclooctyl-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(4-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}phenyl)acetic acid
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
2-benzyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1,3-benzoxazole-5-carboxamide
2-(ethylamino)-N-{2-[methyl(phenyl)amino]propyl}pyrimidine-5-carboxamide
dimethyl({[5-(2-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl})amine
4-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]amino}-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)[2-(pyrrolidin-1-yl)ethyl]amine
(1R,5R)-3-methanesulfonyl-6-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
(3S,4R)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
6-fluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)acetamide
1-cyclohexyl-3-(3-methoxyphenoxymethyl)-5-(oxan-4-yl)-1H-1,2,4-triazole
1-(cyclopropylmethyl)-5-(9H-fluoren-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
N-(1,3-dihydroxy-2-methylpropan-2-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]propanamide
4-{1-cyclohexyl-5-[(1S)-1-(methylamino)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
N-cyclopropyl-7-(quinoline-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-8-methoxyquinoline
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4aS,8aS)-7-(dimethyl-1,3-thiazol-2-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(dimethylamino)ethan-1-one