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1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-2-methyl-1,4-diazepan-5-one
4-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyridine
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methoxypyrimidine
1-benzyl-N-cyclopropyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
N-butyl-1-cyclohexyl-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
2-amino-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-methyl-1,3-benzothiazole-6-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylic acid
3-[3-(3-cyclohexylpyrrolidin-1-yl)propyl]-5-methyl-4H-1,2,4-triazole
N-cyclopentyl-3-[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]propanamide
9-(cyclopropylmethyl)-4-(4-methoxypyrimidin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
5-[({[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
ethyl 4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine-1-carboxylate
ethyl 1-(1-acetylpiperidin-4-yl)-3-benzylpiperidine-3-carboxylate
[2-(1H-imidazol-1-yl)ethyl](methyl)({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)amine
4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)-N-(5-propyl-4H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
8-(1H-1,3-benzodiazol-2-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-1-benzyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
3-(1-ethoxypropyl)-4-(3-methylphenyl)-4H-1,2,4-triazole
1-[2-(methylamino)pyrimidine-5-carbonyl]-N-(2-phenylethyl)piperidine-4-carboxamide
3-({[(2,5-dimethylphenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-(2-ethyl-1H-imidazol-1-yl)acetamide
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
3-{3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]propoxy}pyridine
3-methyl-8-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-methoxy-1-[1'-(3-methoxypyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[3-(5-methylfuran-2-yl)benzoyl]-N-phenylpiperidin-3-amine
[(2S)-1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
3-(2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
methyl (1R,3S,3aR,6aS)-3-[(2E)-but-2-en-2-yl]-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
8-(2,6-diaminopyrimidin-4-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(3-methoxypropyl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
3-(dimethylsulfamoyl)-N-[2-(oxan-2-yl)ethyl]benzamide
[(3S,5R)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-[2-(4-methoxyphenyl)ethyl]-4-pentanamidobenzamide
7-[(2,3-difluorophenyl)methyl]-2-(oxane-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
5-(2-methoxyphenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridine-3-carboxylic acid
1-[1-(4,6-dimethylquinolin-2-yl)piperidin-4-yl]piperidin-3-ol
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-{[(4-methylphenyl)amino]methyl}benzamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-(oxan-4-yl)piperidine-3-carboxamide
N-cyclopropyl-3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}propanamide
1-ethyl-5-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)-1H-1,2,4-triazole
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
2-(hydroxymethyl)-N-[3-(3-methylphenyl)phenyl]azepane-1-carboxamide
N-[2-(naphthalen-1-yl)propan-2-yl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
4-(1-benzothiophen-2-ylmethyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine