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methyl 5-[(2-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamido)methyl]furan-2-carboxylate
(1R,9aR)-1-{[(5-hydroxypentyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
1-[benzyl(methyl)amino]-3-[4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
(3R,5S)-N-butyl-5-(3-fluorophenoxymethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
N-[2-(morpholin-4-yl)ethyl]-4-{4-[(prop-2-en-1-yl)amino]piperidin-1-yl}benzamide
5-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}thiophene-2-carboxylic acid
(1R,2S)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-propylcyclopropane-1-carboxamide
N-benzyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidin-2-amine
7-fluoro-2-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]quinoline-4-carboxamide
1-(pyrimidin-5-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
8-[2-(3-fluorophenoxy)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
5-chloro-2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-phenyl-1H-indole
(3aS,6aR)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(5-methylhex-5-en-2-yl)piperidine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-{7-methyl-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperidin-4-ol
2-ethyl-4-phenyl-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-benzofuran-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
2-[1-(2-methoxyethyl)pyrrolidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(5-chloro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[(2-methyl-4-phenylpiperazin-1-yl)methyl]phenyl}ethan-1-one
N-methyl-N-[2-(methylsulfanyl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-hydroxy-3-phenyl-N-[3-(pyridin-2-yl)propyl]propanamide
N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2-[3-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)propyl]phenol
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-2-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)acetamide
(3R)-3,4,4-trimethyl-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-ol
3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(1H-pyrazol-1-yl)phenyl]urea
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-methoxypyridine-4-carboxamide
5-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-ethyl-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(4-hydroxyphenyl)propyl]-1-methyl-1H-indole-4-carboxamide
6-methyl-N-(propan-2-yl)-5-[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperidin-3-ol
ethyl 1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxylate
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-4,6-dimethylpyridine-3-carbonitrile
3-[5-(1H-1,2,3-benzotriazol-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methoxypyrimidin-4-amine
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-methoxy-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
6-[3-(1-methoxyethyl)phenyl]pyrimidin-4-amine
4-[2-(1-ethylpiperidin-4-yl)acetyl]-1-phenylpiperazine-2-carboxylic acid
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
(1R,3S)-3-{[2-(benzyloxy)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one