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ethyl 5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[(2-fluorophenyl)methyl]piperidine
N-({1-[(2-ethyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
2-ethyl-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)butanamide
N-methyl-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-(piperidin-4-yl)benzamide
(4aS,8aR)-6-[4-(hydroxymethyl)benzoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(2-methyl-1H-indol-3-yl)ethan-1-one
ethyl 4-[3-({[2-(3,4-dimethoxyphenyl)ethyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
N-(2-fluoro-5-methylphenyl)-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane-1-carboxamide
2-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]aniline
5-[(methylsulfanyl)methyl]-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]furan-2-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(propane-2-sulfonyl)piperidine
{5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]furan-2-yl}methanol
1-(3-chlorophenyl)-4-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperazin-2-one
5,5-dimethyl-3-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,3-oxazolidine-2,4-dione
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(oxan-2-yl)ethyl]amine
4-hydroxy-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-1-methylpiperidine-4-carboxamide
2-{[(2,4-dimethoxyphenyl)methyl]amino}-N-(2,3-dimethylphenyl)acetamide
1-{2-[4-(4-chlorophenoxy)piperidine-1-carbonyl]phenyl}ethan-1-one
N-[(2-chlorophenyl)methyl]-3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
4-(3-benzyl-1H-pyrazol-5-yl)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidine
9-[(2-methoxy-4-methylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3,5-dichloro-2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
{3-[(3-chlorophenyl)methyl]-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl}methanol
ethyl 3-benzyl-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxylate
(2R)-2-[5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
N-(2-methoxyethyl)-4-(piperidin-3-yl)-N-(thiophen-3-ylmethyl)benzamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-3-methylpiperidine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}butanamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl[2-methyl-2-(morpholin-4-yl)propyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
2-(dimethylamino)-2-(2-methylphenyl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-(5-chloro-2-methoxybenzoyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
1-[(4-methylphenyl)amino]-N-[(2S)-oxolan-2-ylmethyl]cyclopentane-1-carboxamide
7-(4-chloro-1H-pyrazole-3-carbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[1-(piperidin-1-yl)cyclohexyl]methyl}amine
propan-2-yl 8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
N-(pyridin-4-ylmethyl)-4-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(3-{[methyl(1,2-oxazol-3-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
4-(3,6-dimethylpyrazin-2-yl)-1H-indole
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
8-(6-methoxypyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(3-cyclopentylpropyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{3-[1-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]propyl}dimethylamine
1-{6-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperazin-1-yl]pyridin-3-yl}ethan-1-one
(1R,5S)-3-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane