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(cyclohex-1-en-1-ylmethyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
3-(1H-imidazol-1-ylmethyl)-N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}piperidine-1-carboxamide
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-amino-N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-4-methyl-1,3-benzothiazole-6-carboxamide
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
methyl 5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-aminoethyl)-4-[3-(methylsulfanyl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decane
2-(2-hydroxyethyl)-8-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
methyl 3-{[(2-hydroxyethyl)[(2-methoxyphenyl)methyl]carbamoyl]amino}-4-methylbenzoate
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-methylacetamide
3-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-2,6-dimethyl-1,4-dihydropyridin-4-one
2-[(5-phenylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1s,4s)-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
(3S,4R)-4-methyl-1-[4-(morpholine-4-carbonyl)benzoyl]piperidine-3,4-diol
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
2-benzyl-6-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-({1-[(2,3-dimethyl-1H-indol-7-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
1-(2-{[2-(2-methoxyphenyl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
4-chloro-1-ethyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazole
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
N-({5-[(2,2-dimethyloxan-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1-{3-[(5-ethylpyrimidin-2-yl)amino]propyl}piperidin-3-yl)methanol
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
5-ethyl-2-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-phenylphenyl)methyl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
N-cyclopropyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-(methoxymethyl)-N-[2-(2-methoxyphenoxy)ethyl]cyclobutane-1-carboxamide
N4-[(2,4-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-(4-chlorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)cyclobutane-1-carboxamide
ethyl 1-(cyclopropylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-methylcyclohexanecarbonyl)piperidin-3-ol
2-[(4-chlorophenyl)methyl]-8-(5-methyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidine-4-carboxamide
2-[3-(dimethylamino)propyl]-9-[2-(3-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(methoxymethyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-chloro-N-(2-hydroxypropyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-[(2-methylpropyl)amino]benzamide
3-[3-(4-methoxyphenyl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2,2,2-trifluoroethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-benzyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
2-[1-(3-methylphenyl)-5-{[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-3-yl]acetamide
2-[(3-{[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
1-methyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole